SCHEMBL9024624

SCHEMBL9024624

COC(=O)COc1[c]cc(Cl)cc1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.50
LMNA P02545 1/20 0.45
PTGDR Q13258 1/20 0.43
PTGDR2 Q9Y5Y4 1/20 0.43
CYP1A2 P05177 3/20 0.40
CYP2C9 P11712 1/20 0.40
HIF1A Q16665 1/20 0.40
KMT2A Q03164 3/20 0.40
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.39
MEN1 O00255 2/20 0.38
ALDH1A1 P00352 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
LPAR2 Q9HBW0 1/20 0.35
BLM P54132 1/20 0.35
PMP22 Q01453 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL324953 0.81 TDP1 (0.49) PTGDRPTGDR2KMT2AMAPTALDH1A1
SCHEMBL9023430 0.81 HPGD (0.40) PTGS2LMNACYP1A2CYP2C9KMT2A
SCHEMBL9024232 0.78 SMN1; SMN2 (0.41) PTGS2LMNACYP1A2KMT2AMAPT
SCHEMBL9024894 0.77 PPARG (0.43) LMNACYP1A2CYP2C9KMT2AKDM4E
SCHEMBL9024538 0.77 ALDH1A1 (0.46) LMNACYP1A2CYP2C9KMT2AKDM4E
SCHEMBL9023743 0.74 LMNA (0.53) PTGS2LMNAPTGDRPTGDR2CYP1A2
SCHEMBL9111454 0.74 PTPN1 (0.32)
SCHEMBL5120243 0.74 PTGS2 (0.81) PTGS2LMNACYP1A2CYP2C9KMT2A
SCHEMBL2565533 0.73 KMT2A (0.40) PTGS2LMNACYP1A2KMT2AKDM4E
SCHEMBL162984 0.73 NQO1 (0.36) LMNAKMT2AKDM4EMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0398179-B1 Rhodanine derivatives and pharmaceutical compositions NISSHIN FLOUR MILLING CO (JP) 1996-01-17 EP disclosed
US-5116855-A Aldose reductase inhibitors; antidiabetic agents NISSHIN FLOUR MILLING CO., LTD. (JP) 1992-05-26 US disclosed
EP-0398179-A1 Rhodanine derivatives and pharmaceutical compositions NISSHIN FLOUR MILLING CO., LTD. (JP) 1990-11-22 EP disclosed