SCHEMBL9026027

SCHEMBL9026027

CCOc1ccc(Cl)cc1N(C)c1occ2ccccc12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.35
HPGD P15428 1/20 0.35
HTR2C P28335 2/20 0.34
HTR2B P41595 2/20 0.34
HTR2A P28223 1/20 0.34
ALOX5 P09917 1/20 0.34
POLB P06746 2/20 0.34
THRB P10828 2/20 0.34
LMNA P02545 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HTT P42858 1/20 0.34
MAPT P10636 1/20 0.34
TP53 P04637 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
SLC2A1 P11166 1/20 0.34
AGPAT2 O15120 1/20 0.33
ENPP1 P22413 1/20 0.33
ATM Q13315 1/20 0.33
S1PR1 P21453 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9025560 0.86 METAP2 (0.40) TSHRPOLBALDH1A1HTTMAPT
SCHEMBL9032006 0.83 CYP1A2 (0.36) POLBHTTMAPTCYP1A2ATM
SCHEMBL9026425 0.81 TSHR (0.35) TSHRHPGDHTR2CHTR2BHTR2A
SCHEMBL9025461 0.80 TP53 (0.35) TSHRHPGDHTR2APOLBLMNA
SCHEMBL9025423 0.79 HSD17B10 (0.34) TSHRHPGDMAPTCYP1A2CYP2D6
SCHEMBL9025676 0.74 ACLY (0.41) TSHRLMNAHTTMAPTMAPK1
SCHEMBL9025102 0.73 MAPK1 (0.37) TSHRPOLBLMNAHTTMAPT
SCHEMBL9026853 0.73 GAA (0.45) TSHRHPGDPOLBLMNAALDH1A1
SCHEMBL9025513 0.73 ALDH1A1 (0.50) TSHRHPGDPOLBLMNAALDH1A1
SCHEMBL9026655 0.72 GLA (0.36) TSHRHTR2CHTR2BHTR2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0711290-A1 METHYLGUANIDINE DERIVATIVES, METHODS FOR PREPARING SAME AND COMPOSITIONS CONTAINING SAID DERIVATIVES SANOFI (FR) 1996-05-15 EP disclosed
WO-1995004052-A1 METHYLGUANIDINE DERIVATIVES, METHODS FOR PREPARING SAME AND COMPOSITIONS CONTAINING SAID DERIVATIVES SANOFI (FR) 1995-02-09 WO disclosed