SCHEMBL9032006

SCHEMBL9032006

CC(C)Oc1ccc(Cl)cc1N(C)c1occ2ccccc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.36
MAPT P10636 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
METAP2 P50579 1/20 0.33
ATM Q13315 1/20 0.33
TSPO P30536 1/20 0.32
SHMT2 P34897 1/20 0.32
MAP2 P11137 1/20 0.32
TLR8 Q9NR97 1/20 0.32
NPC1 O15118 2/20 0.31
KMT2A Q03164 2/20 0.31
MEN1 O00255 1/20 0.31
POLB P06746 1/20 0.31
HTT P42858 1/20 0.31
IRAK4 Q9NWZ3 1/20 0.31
RAB9A P51151 1/20 0.30
ADORA3 P0DMS8 1/20 0.30
SLC9A1 P19634 1/20 0.30
S1PR1 P21453 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9025560 0.86 METAP2 (0.40) MAPTMETAP2SHMT2NPC1KMT2A
SCHEMBL9026027 0.83 TSHR (0.35) CYP1A2MAPTATMPOLBHTT
SCHEMBL9026534 0.82 SLC9A1 (0.35) CYP1A2MAPTCYP2C9CYP2C19TSPO
SCHEMBL9025461 0.80 TP53 (0.35) CYP1A2MAPTNPC1KMT2AMEN1
SCHEMBL9025423 0.79 HSD17B10 (0.34) CYP1A2MAPTCYP2C9CYP2C19KMT2A
SCHEMBL9025676 0.74 ACLY (0.41) MAPTSHMT2NPC1KMT2AMEN1
SCHEMBL9026853 0.73 GAA (0.45) CYP1A2MAPTNPC1KMT2AMEN1
SCHEMBL9025513 0.73 ALDH1A1 (0.50) MAPTMETAP2KMT2AMEN1POLB
SCHEMBL9026655 0.72 GLA (0.36) MAPTSHMT2KMT2AMEN1POLB
SCHEMBL9024891 0.72 NQO1 (0.37) MAPTNPC1KMT2AMEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0711290-A1 METHYLGUANIDINE DERIVATIVES, METHODS FOR PREPARING SAME AND COMPOSITIONS CONTAINING SAID DERIVATIVES SANOFI (FR) 1996-05-15 EP disclosed
WO-1995004052-A1 METHYLGUANIDINE DERIVATIVES, METHODS FOR PREPARING SAME AND COMPOSITIONS CONTAINING SAID DERIVATIVES SANOFI (FR) 1995-02-09 WO disclosed