SCHEMBL9026327

SCHEMBL9026327

COc1ccc(-c2cccnc2)cc1N(C)c1occ2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 6/20 0.47
CYP11B1 P15538 5/20 0.47
CYP19A1 P11511 4/20 0.47
CYP17A1 P05093 3/20 0.43
NPC1 O15118 4/20 0.42
RAB9A P51151 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
MAPT P10636 4/20 0.42
KDM4E B2RXH2 1/20 0.41
MAPK1 P28482 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TLR8 Q9NR97 2/20 0.41
TLR7 Q9NYK1 2/20 0.41
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
ALDH1A1 P00352 2/20 0.41
ABCB1 P08183 3/20 0.40
ABCC1 P33527 2/20 0.40
PDGFRB P09619 1/20 0.40
PDGFRA P16234 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9032013 0.88 MAPT (0.37) CYP17A1NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL9025511 0.82 KDM4E (0.38) NPC1RAB9ASMN1; SMN2MAPTKDM4E
SCHEMBL9026853 0.78 GAA (0.45) NPC1RAB9ASMN1; SMN2MAPTKDM4E
SCHEMBL9025513 0.78 ALDH1A1 (0.50) MAPTKDM4EHSD17B10ALDH1A1PDGFRB
SCHEMBL9025554 0.77 MAPK14 (0.39) MAPTKDM4EMAPK1ALDH1A1ABCB1
SCHEMBL9024891 0.77 NQO1 (0.37) NPC1RAB9ASMN1; SMN2MAPTKDM4E
SCHEMBL9025087 0.77 ALDH1A1 (0.39) NPC1RAB9ASMN1; SMN2MAPTKDM4E
SCHEMBL9026004 0.77 NQO1 (0.37) MAPTALDH1A1GAA
SCHEMBL9216015 0.77 NQO1 (0.37) MAPTALDH1A1PDGFRBGAA
SCHEMBL9025560 0.77 METAP2 (0.40) NPC1RAB9ASMN1; SMN2MAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0711290-A1 METHYLGUANIDINE DERIVATIVES, METHODS FOR PREPARING SAME AND COMPOSITIONS CONTAINING SAID DERIVATIVES SANOFI (FR) 1996-05-15 EP disclosed
WO-1995004052-A1 METHYLGUANIDINE DERIVATIVES, METHODS FOR PREPARING SAME AND COMPOSITIONS CONTAINING SAID DERIVATIVES SANOFI (FR) 1995-02-09 WO disclosed