SCHEMBL9026464

SCHEMBL9026464

COc1ccc(Oc2ccccc2)cc1C(N)c1occ2ccccc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.39
NQO1 P15559 1/20 0.37
ADRA2A P08913 2/20 0.36
ADRA1A P35348 2/20 0.36
CYP2D6 P10635 1/20 0.36
MAPT P10636 2/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
MAPK1 P28482 1/20 0.35
BLM P54132 1/20 0.35
TSPO P30536 1/20 0.35
GPR84 Q9NQS5 2/20 0.34
HCRTR1 O43613 1/20 0.34
HCRTR2 O43614 1/20 0.34
LMNA P02545 3/20 0.34
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 2/20 0.34
HTT P42858 2/20 0.34
HPGD P15428 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9026859 0.90 ADRA2A (0.45) NQO1ADRA2AADRA1ACYP2D6MAPT
SCHEMBL9025520 0.83 METAP2 (0.38) NQO1MAPTMEN1KMT2AGPR84
SCHEMBL9025089 0.83 KDM4E (0.41) NQO1MAPTMEN1KMT2AMAPK1
SCHEMBL9026008 0.82 PKM (0.38) NQO1MAPTGPR84
SCHEMBL9216019 0.82 NQO1 (0.36) NQO1MAPTGPR84
SCHEMBL9024896 0.82 MYB (0.36) NQO1MAPTMEN1KMT2AGPR84
SCHEMBL9025436 0.79 TSHR (0.39) MEN1KMT2AMAPK1GPR84HCRTR1
SCHEMBL9026458 0.76 KDM4E (0.41) LTA4HADRA2AADRA1ACYP2D6MAPT
SCHEMBL9025514 0.76 PDE4A (0.39) MAPTMEN1KMT2ALMNAKDM4E
SCHEMBL9026660 0.75 MAPT (0.35) NQO1MAPTMEN1KMT2AGPR84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0711290-A1 METHYLGUANIDINE DERIVATIVES, METHODS FOR PREPARING SAME AND COMPOSITIONS CONTAINING SAID DERIVATIVES SANOFI (FR) 1996-05-15 EP disclosed
WO-1995004052-A1 METHYLGUANIDINE DERIVATIVES, METHODS FOR PREPARING SAME AND COMPOSITIONS CONTAINING SAID DERIVATIVES SANOFI (FR) 1995-02-09 WO disclosed