SCHEMBL9216019

SCHEMBL9216019

COc1ccc(I)cc1C(N)c1occ2ccccc12

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 1/20 0.36
MAPT P10636 1/20 0.35
GPR84 Q9NQS5 1/20 0.34
IDO1 P14902 2/20 0.33
BCHE P06276 2/20 0.33
ACHE P22303 2/20 0.33
SOS1 Q07889 5/20 0.32
KRAS P01116 4/20 0.32
MYB P10242 1/20 0.32
EGFR P00533 1/20 0.32
APP P05067 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9025520 0.86 METAP2 (0.38) NQO1MAPTGPR84ACHEMYB
SCHEMBL9025089 0.86 KDM4E (0.41) NQO1MAPTGPR84
SCHEMBL9026859 0.86 ADRA2A (0.45) NQO1MAPTACHE
SCHEMBL9026008 0.85 PKM (0.38) NQO1MAPTGPR84IDO1ACHE
SCHEMBL9025568 0.85 METAP2 (0.39) NQO1MAPTGPR84ACHE
SCHEMBL9024896 0.85 MYB (0.36) NQO1MAPTGPR84ACHEMYB
SCHEMBL9026464 0.82 LTA4H (0.39) NQO1MAPTGPR84
SCHEMBL9032018 0.80 DHFR (0.39) MAPT
SCHEMBL9025436 0.79 TSHR (0.39) GPR84
SCHEMBL9025514 0.78 PDE4A (0.39) MAPTSOS1KRAS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995004052-A1 METHYLGUANIDINE DERIVATIVES, METHODS FOR PREPARING SAME AND COMPOSITIONS CONTAINING SAID DERIVATIVES SANOFI (FR) 1995-02-09 WO claimed
WO-1995004052-A1 METHYLGUANIDINE DERIVATIVES, METHODS FOR PREPARING SAME AND COMPOSITIONS CONTAINING SAID DERIVATIVES SANOFI (FR) 1995-02-09 WO disclosed