SCHEMBL904087

SCHEMBL904087

CS(=O)(=O)c1ccc(-c2ccc(O)c(Cl)c2)cc1

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 2/20 0.56
PTGS2 P35354 12/20 0.50
ENPP2 Q13822 1/20 0.48
ESR1 P03372 1/20 0.47
ACLY P53396 1/20 0.47
PTGS1 P23219 1/20 0.47
HSD17B1 P14061 2/20 0.45
HSD17B2 P37059 2/20 0.45
HDAC2 Q92769 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1577287 0.85 LMNA (0.55) PTGS2ENPP2ACLYPTGS1HSD17B2
SCHEMBL5715742 0.83 APP (0.56) PTGS2ENPP2
SCHEMBL6513992 0.82 ENPP2 (0.64) PTGS2ENPP2PTGS1HSD17B2
SCHEMBL10068013 0.80 HSD17B1 (0.53) ESR2PTGS2ENPP2ESR1HSD17B1
SCHEMBL8055957 0.79 PTGS2 (0.77) PTGS2PTGS1
SCHEMBL386673 0.79 KIF11 (0.61) ESR2PTGS2ENPP2ESR1PTGS1
SCHEMBL28184683 0.78 AVPR2 (0.50) PTGS2PTGS1
SCHEMBL28202577 0.78 ESR2 (0.77) ESR2ESR1HSD17B1HSD17B2HDAC2
SCHEMBL278316 0.78 ESR2 (0.77) ESR2ESR1HSD17B1HSD17B2HDAC2
SCHEMBL29911026 0.78 ESR2 (0.77) ESR2ESR1HSD17B1HSD17B2HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102432598-A Tricyclic compound, preparation method thereof and pharmaceutical application thereof JIANGSU HENGRUI MEDICINE CO 2012-05-02 CN disclosed
WO-2012041158-A1 TRICYCLIC COMPOUND, PREPARATION METHOD AND PHARMACEUTICAL USE THEREOF 上海恒瑞医药有限公司 (CN) 2012-04-05 WO disclosed