SCHEMBL9044348

SCHEMBL9044348

O=C(CNC(=O)OCc1ccccc1)N[C@@H](Cc1ccccc1)C(=O)ON1C(=O)CCC1=O

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.47
CTSL P07711 4/20 0.46
CTSB P07858 3/20 0.46
CTSS P25774 1/20 0.46
CTSK P43235 1/20 0.46
CASP1 P29466 1/20 0.46
CYP3A4 P08684 1/20 0.46
TYR P14679 1/20 0.45
TACR1 P25103 3/20 0.44
ACE P12821 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17039822 0.89 TACR1 (0.55) ALDH1A1CTSLCTSBCTSSCTSK
SCHEMBL5689118 0.89 TACR1 (0.55) ALDH1A1CTSLCTSBCTSSCTSK
SCHEMBL14488100 0.89 TACR1 (0.55) ALDH1A1CTSLCTSBCTSSCTSK
SCHEMBL29973202 0.87 KLK5 (0.50) CTSLCTSBCTSSCTSKACE
SCHEMBL30971331 0.86 CASP1 (0.44) ALDH1A1CASP1TACR1
SCHEMBL8208600 0.85 CTSB (0.56) ALDH1A1CTSLCTSBCTSSCTSK
SCHEMBL31418693 0.83 ALDH1A1 (0.51) ALDH1A1CASP1
SCHEMBL5352301 0.83 ALDH1A1 (0.51) ALDH1A1CASP1
SCHEMBL30442090 0.83 ALDH1A1 (0.51) ALDH1A1CASP1
SCHEMBL25148105 0.83 OPRD1 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0360258-B1 Amino acid quinoline and naphthyridine derivatives ABBOTT LAB (US) 1996-08-14 EP disclosed
US-5057523-A Water soluble bactericide ABBOTT LABORATORIES (US) 1991-10-15 US disclosed
US-5057520-A Water solubility ABBOTT LABORATORIES (US) 1991-10-15 US disclosed
EP-0360258-A2 Amino acid quinoline and naphthyridine derivatives ABBOTT LABORATORIES (US) 1990-03-28 EP disclosed
EP-0295316-A2 Antitumor amino acid and peptide derivatives of 1,4-bis[ (aminoalkyl and hydroxyaminoalkyl)- amino]-5,8 dihydroxyanthraquinones AMERICAN CYANAMID COMPANY (US) 1988-12-21 EP disclosed
US-4732970-A Antitumor amino acid and peptide derivatives of 1,4-bis(aminoalkyl and hydroxy-aminoalkyl)amino)-5,8-dihydroxyanthraquinones AMERICAN CYANAMID COMPANY (US) 1988-03-22 US disclosed