SCHEMBL9047265

SCHEMBL9047265

O=C(O)c1cn(-c2ccon2)c2cc(F)c(F)c(Cl)c2c1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
HTT P42858 1/20 0.40
STAT3 P40763 1/20 0.38
TOP1 P11387 2/20 0.35
CHRM1 P11229 3/20 0.33
KDM4E B2RXH2 2/20 0.33
POLB P06746 1/20 0.33
HSP90AA1 P07900 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
LMNA P02545 2/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
PIM1 P11309 1/20 0.32
HPGD P15428 1/20 0.32
HSD17B10 Q99714 1/20 0.32
GAA P10253 1/20 0.32
CYP3A4 P08684 3/20 0.31
RORC P51449 1/20 0.31
CYP2C9 P11712 2/20 0.31
GSK3B P49841 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9047564 0.89 ALDH1A1 (0.40) ALDH1A1HTTSTAT3TOP1CHRM1
SCHEMBL9044750 0.88 ALDH1A1 (0.41) ALDH1A1HTTSTAT3TOP1CHRM1
SCHEMBL9045879 0.87 ALDH1A1 (0.40) ALDH1A1HTTSTAT3TOP1KDM4E
SCHEMBL9045934 0.85 HTT (0.46) ALDH1A1HTTSTAT3KDM4ELMNA
SCHEMBL9047248 0.83 ALDH1A1 (0.40) ALDH1A1HTTSTAT3TOP1KDM4E
SCHEMBL9048751 0.83 TOP1 (0.45) ALDH1A1HTTTOP1CHRM1KDM4E
SCHEMBL9045282 0.81 LMNA (0.43) ALDH1A1HTTTOP1KDM4EPOLB
SCHEMBL9046944 0.76 ALDH1A1 (0.53) ALDH1A1HTTSTAT3TOP1KDM4E
SCHEMBL9046043 0.74 STAT3 (0.54) ALDH1A1HTTSTAT3TOP1CHRM1
SCHEMBL9047636 0.73 HTT (0.46) ALDH1A1HTTSTAT3KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0700912-A1 QUINOLONE DERIVATIVE OR SALT THEREOF, AND ANTIBACTERIAL CONTAINING THE SAME WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1996-03-13 EP disclosed