SCHEMBL9057955

SCHEMBL9057955

O=C(O)c1n[nH]c(-c2ccccc2)c1Br

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.47
LMNA P02545 1/20 0.47
TP53 P04637 1/20 0.42
HCAR2 Q8TDS4 2/20 0.41
MAPK1 P28482 2/20 0.41
PIN1 Q13526 2/20 0.41
CYP1A2 P05177 1/20 0.41
CASP1 P29466 1/20 0.41
CYP2C19 P33261 1/20 0.41
ALDH1A1 P00352 4/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
GAA P10253 2/20 0.41
HPGD P15428 2/20 0.41
HSD17B10 Q99714 2/20 0.41
DYRK1B Q9Y463 2/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
PLA2G10 O15496 1/20 0.39
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29408204 0.81 PRKAG1 (0.56) KDM4ELMNATP53CYP1A2CYP2C19
SCHEMBL570062 0.79 PIN1 (0.47) KDM4ELMNATP53HCAR2MAPK1
SCHEMBL11622011 0.75 KDM4E (0.47) KDM4ETP53MAPK1ALDH1A1SMN1; SMN2
SCHEMBL10642212 0.75 LMNA (0.44) KDM4ELMNATP53MAPK1PIN1
SCHEMBL8887039 0.73 ALDH1A1 (0.60) KDM4ELMNATP53MAPK1CYP1A2
SCHEMBL2875437 0.72 MAPK1 (0.63) KDM4ETP53MAPK1CYP1A2CYP2C19
SCHEMBL16225421 0.72 AKT2 (0.50) KDM4ETP53MAPK1ALDH1A1SMN1; SMN2
SCHEMBL15799669 0.71 ALPL (0.48) KDM4ELMNATP53HCAR2MAPK1
SCHEMBL20028652 0.70 KDM4E (0.46) KDM4ELMNATP53MAPK1PIN1
SCHEMBL2198685 0.70 IKBKB (0.43) KDM4EHCAR2MAPK1PIN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996012706-A1 NOVEL ACID PYRAZOLE AND PYRAZOLONE DERIVATIVES FOR USE AS ENDOTHELIN RECEPTOR ANTAGONISTS ROUSSEL UCLAF (FR) 1996-05-02 WO disclosed