SCHEMBL91304

SCHEMBL91304

CCOOCC1=C(OS(=O)(=O)C(F)(F)F)CC(CCC(C)(C)[Si](C)(C)O)N(C(=O)OCc2ccccc2)C1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.35
PDK2 Q15119 1/20 0.35
PDK3 Q15120 1/20 0.35
PDK4 Q16654 1/20 0.35
CCR5 P51681 1/20 0.33
HTR2C P28335 1/20 0.32
PTPN1 P18031 1/20 0.32
RORC P51449 1/20 0.32
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
TSHR P16473 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
KDM4E B2RXH2 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL91250 0.82 PARP1 (0.34) PDK1PDK2PDK3PDK4CCR5
SCHEMBL91259 0.80 HTR2C (0.33) PDK1PDK2PDK3PDK4HTR2C
SCHEMBL78407 0.79 PDK1 (0.37) PDK1PDK2PDK3PDK4CCR5
SCHEMBL91189 0.77 PDK1 (0.36) PDK1PDK2PDK3PDK4CCR5
SCHEMBL14420341 0.77 HTR2C (0.41) PDK1PDK2PDK3PDK4HTR2C
SCHEMBL91296 0.76 PDK1 (0.36) PDK1PDK2PDK3PDK4HTR2C
SCHEMBL64675 0.75 PDK1 (0.38) PDK1PDK2PDK3PDK4CCR5
SCHEMBL91275 0.74 PPARG (0.38) ALDH1A1TSHRL3MBTL1KDM4ELMNA
SCHEMBL91257 0.74 ITGB3 (0.34) KDM4ELMNA
SCHEMBL78189 0.73 PDK1 (0.38) PDK1PDK2PDK3PDK4CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129538-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-06 US disclosed