SCHEMBL9130874

SCHEMBL9130874

COC(=O)CCCCCCN1CCN(c2nc(N3CCCC3)nc(N3CCCC3)c2OC(=O)c2ccccc2)CC1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 8/20 0.42
DRD2 P14416 6/20 0.42
HTR7 P34969 4/20 0.41
DRD3 P35462 3/20 0.41
HTR2A P28223 2/20 0.41
HTR6 P50406 1/20 0.41
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HTT P42858 1/20 0.40
DRD4 P21917 2/20 0.39
SIGMAR1 Q99720 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9756683 0.84 CASP1 (0.43) HTR1ADRD2KDM4EALDH1A1HTT
SCHEMBL9131819 0.77 CASP1 (0.50)
SCHEMBL9690061 0.76 CASP1 (0.51)
SCHEMBL9671054 0.74 ALDH1A1 (0.46) ALDH1A1SIGMAR1
SCHEMBL1085753 0.74 HTR1A (0.65) HTR1ADRD2HTR7DRD3HTR2A
SCHEMBL9756638 0.73 GBA1 (0.49)
SCHEMBL9689589 0.72 CASP1 (0.47)
SCHEMBL29183995 0.69 DRD2 (0.43) HTR1ADRD2HTR7DRD3HTR6
SCHEMBL29183819 0.69 PIK3CA (0.60)
SCHEMBL28390299 0.68 PAOX (0.53) HTR1AHTR7ALDH1A1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992018089-A2 USE OF STEROIDAL AND NON-STEROIDAL AMINES TO SENSITIZE MULTIDRUG-RESISTANT CELLS THE UPJOHN COMPANY (US) 1992-10-29 WO claimed
US-5436337-A Anticarcinogenic agents THE UPJOHN COMPANY (US) 1995-07-25 US disclosed
WO-1992018089-A2 USE OF STEROIDAL AND NON-STEROIDAL AMINES TO SENSITIZE MULTIDRUG-RESISTANT CELLS THE UPJOHN COMPANY (US) 1992-10-29 WO disclosed