SCHEMBL9199668

SCHEMBL9199668

O=C1CCC2(CC1)CC(O)=C(CCCc1ccccc1)C(=O)O2

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XIAP P98170 1/20 0.37
TSHR P16473 2/20 0.36
LMNA P02545 1/20 0.36
CHRM2 P08172 1/20 0.36
ADRA2A P08913 1/20 0.36
CYP2D6 P10635 1/20 0.36
DRD1 P21728 1/20 0.36
KMT2A Q03164 2/20 0.36
MAPT P10636 1/20 0.36
DRD2 P14416 2/20 0.36
SIGMAR1 Q99720 1/20 0.36
ESR1 P03372 1/20 0.35
ESR2 Q92731 1/20 0.35
TAAR1 Q96RJ0 2/20 0.34
HSD11B1 P28845 2/20 0.34
HTR2A P28223 1/20 0.34
HTR2B P41595 1/20 0.34
NR3C1 P04150 1/20 0.34
AR P10275 1/20 0.34
HDAC3 O15379 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9198495 0.88 ALDH1A1 (0.39) XIAPTSHRLMNACHRM2ADRA2A
SCHEMBL9195252 0.85 HSD11B1 (0.38) XIAPTSHRLMNACHRM2ADRA2A
SCHEMBL9199610 0.79 XIAP (0.40) XIAPLMNAMAPTHTR2AHTR2B
SCHEMBL6606184 0.77 LDHA (0.45) XIAPLMNASIGMAR1HTR2BHDAC3
SCHEMBL6175910 0.75 HSD11B1 (0.44) KMT2AHSD11B1MEN1CYP2C9
SCHEMBL9195240 0.72 LDHA (0.38) XIAPESR1ESR2
SCHEMBL9199838 0.71 GAA (0.35) XIAPLMNACHRM2ADRA2ACYP2D6
SCHEMBL6603207 0.69 LDHA (0.47) XIAPTSHRLMNACHRM2ADRA2A
SCHEMBL6175954 0.68 HSD11B1 (0.48) TSHRCHRM2ADRA2ADRD1KMT2A
SCHEMBL8986018 0.66 OPRM1 (0.50) KMT2AMAPTSIGMAR1HDAC3MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0668860-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES PHARMACIA & UPJOHN COMPANY (US) 1995-08-30 EP claimed
EP-0668860-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES PHARMACIA & UPJOHN COMPANY (US) 1995-08-30 EP disclosed