SCHEMBL9204526

SCHEMBL9204526

Cc1cc2c(cc1C)C(=O)N(CCCC1CCCN(CCc3cccc4ccccc34)C1)CC2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
TSHR P16473 1/20 0.38
ADRA1D P25100 2/20 0.37
ADRA1A P35348 2/20 0.37
ADRA1B P35368 2/20 0.37
CHRNB2 P17787 1/20 0.37
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
CHRNA4 P43681 1/20 0.37
SLC18A2 Q05940 1/20 0.37
HTR1A P08908 1/20 0.37
SLC6A4 P31645 1/20 0.37
CXCR4 P61073 1/20 0.37
HDAC3 O15379 2/20 0.36
HDAC4 P56524 2/20 0.36
HDAC1 Q13547 2/20 0.36
HDAC7 Q8WUI4 2/20 0.36
HDAC2 Q92769 2/20 0.36
HDAC10 Q969S8 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9212783 0.88 ADRA1D (0.37) ADRA1DADRA1AADRA1BCHRNB2CHRNB4
SCHEMBL9740802 0.84 SIGMAR1 (0.45) CHRNB2CHRNB4CHRNA3CHRNA4SIGMAR1
SCHEMBL9216594 0.80 PRMT5 (0.39) TSHR
Hydrochloric Acid SCHEMBL9214810 0.79 ADRA1B (0.46) MEN1KMT2AADRA1BCHRNB2CHRNB4
SCHEMBL9213748 0.78 ABCB1 (0.38) TSHR
SCHEMBL10523499 0.78 HDAC3 (0.44) ADRA1DADRA1AADRA1BSLC6A4HDAC3
SCHEMBL9740331 0.78 HRH3 (0.51) MEN1KMT2AHTR1ASLC6A4HRH3
SCHEMBL9217306 0.78 ADRA1B (0.46) MEN1KMT2AADRA1BHTR1ASLC6A4
SCHEMBL9209429 0.77 ADRA1B (0.45) MEN1KMT2AADRA1BHTR1ASLC6A4
SCHEMBL9739974 0.77 HRH3 (0.54) MEN1KMT2AHTR1ASLC6A4HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed