SCHEMBL92056

SCHEMBL92056

[C-]#[N+]c1ccc(-c2ccccc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.50
TAAR1 Q96RJ0 2/20 0.43
CYP1A2 P05177 2/20 0.43
MAPK1 P28482 1/20 0.43
CYP3A4 P08684 1/20 0.43
HSD17B10 Q99714 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
MMP3 P08254 1/20 0.43
BCL2L1 Q07817 1/20 0.43
CTRC Q99895 1/20 0.39
CA1 P00915 4/20 0.39
CA2 P00918 3/20 0.39
MGLL Q99685 2/20 0.39
KIF11 P52732 1/20 0.39
NOTUM Q6P988 1/20 0.38
ALOX5 P09917 1/20 0.37
CA9 Q16790 2/20 0.37
HSD17B3 P37058 1/20 0.37
CYP1A1 P04798 1/20 0.36
CYP1B1 Q16678 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL717099 0.88 EGLN1 (0.34) ALDH1A1CYP3A4TDP1
Biphenyl SCHEMBL11354502 0.84 MMP3 (0.58) ALDH1A1TDP1MMP3BCL2L1CA1
SCHEMBL244994 0.82
SCHEMBL31148860 0.79
SCHEMBL1810851 0.79 CA4 (0.35) ALDH1A1TDP1CA1CA2CA9
SCHEMBL1807521 0.79 CA4 (0.35) ALDH1A1CYP1A2TDP1CA1CA2
Hydrochloric Acid SCHEMBL1304764 0.79 CA4 (0.35) ALDH1A1TDP1CA1CA2CA9
SCHEMBL3734578 0.79 CA4 (0.35) ALDH1A1TDP1CA1CA2CA9
SCHEMBL5589968 0.79 CA4 (0.35) ALDH1A1TDP1CA1CA2CA9
SCHEMBL13019496 0.79 RAB9A (0.60) ALDH1A1MAPK1TDP1CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 34 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114014838-B Compound and preparation method and application thereof 山东师范大学 2024-03-19 CN claimed
CN-113956232-B Quinoline-bisindole compound and preparation method and application thereof 山东师范大学 2022-09-16 CN claimed
CN-114014838-A Compound and preparation method and application thereof 山东师范大学 2022-02-08 CN claimed
CN-113956232-A Quinoline-bisindole compound and preparation method and application thereof 山东师范大学 2022-01-21 CN claimed
CN-118772206-A Isocyanorhodium (I) zwitterionic complex, preparation method thereof, micelle, nano diagnosis and treatment probe and anticancer drug 兰州大学 2024-10-15 CN disclosed
CN-114014838-B Compound and preparation method and application thereof 山东师范大学 2024-03-19 CN disclosed
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
CN-113956232-B Quinoline-bisindole compound and preparation method and application thereof 山东师范大学 2022-09-16 CN disclosed
CN-114014838-A Compound and preparation method and application thereof 山东师范大学 2022-02-08 CN disclosed
CN-113956232-A Quinoline-bisindole compound and preparation method and application thereof 山东师范大学 2022-01-21 CN disclosed
US-20170174582-A1 METHOD FOR COUPLING A FIRST AROMATIC COMPOUND TO A SECOND AROMATIC COMPOUND DOW AGROSCIENCES LLC 2017-06-22 US disclosed
US-9624193-B2 Cyclic azine derivatives, processes for producing these, and organic electroluminescent element containing these as component TOSOH CORPORATION (JP) 2017-04-18 US disclosed
US-8212056-B2 Ligands for transition-metals and methods of use THE HONG KONG POLYTECHNIC UNIVERSITY (CN) 2012-07-03 US disclosed
US-8128848-B2 Diketopyrrolopyrrole pigment composition for use in color filters CLARIANT FINANCE (BVI) LIMITED (VG) 2012-03-06 US disclosed
US-20110046380-A1 METHOD FOR PRODUCING UNSATURATED ORGANIC COMPOUND SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2011-02-24 US disclosed
US-20110028718-A1 PARACYCLOPHANE-BASED LIGANDS, THEIR PREPARATION AND USE IN CATALYSIS JOHNSON MATTHEY PUBLIC LIMITED COMPANY (GB) 2011-02-03 US disclosed
US-20100219384-A1 Diketopyrrolopyrrole Pigment Composition For Use In Color Filters CLARIANT FINANCE (BVI) LIMITED (VG) 2010-09-02 US disclosed
US-20090326243-A1 Ligands for transition-metals and methods of use THE HONG KONG POLYTECHNIC UNIVERSITY (HK) 2009-12-31 US disclosed
US-7534894-B2 Biphenyloxy-acids WYETH (US) 2009-05-19 US disclosed
US-7332499-B2 Sulfonyl substituted n-(biarylmethyl) aminocyclopropanecarboxamides MERCK & CO., INC. (US) 2008-02-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110028718-A1 PARACYCLOPHANE-BASED LIGANDS, THEIR PREPARATION AND USE IN CATALYSIS C1S, XDH, CYCS ALDH1A1 2148/4885TAAR1 1342/4885CYP1A2 22/4885
US-20170174582-A1 METHOD FOR COUPLING A FIRST AROMATIC COMPOUND TO A SECOND AROMATIC COMPOUND PAH, TYR, AHR ALDH1A1 1437/4885TAAR1 724/4885CYP1A2 320/4885
US-20090326243-A1 Ligands for transition-metals and methods of use PDK4, PDXK, PDK3 ALDH1A1 1267/4885TAAR1 1450/4885CYP1A2 776/4885
US-20110046380-A1 METHOD FOR PRODUCING UNSATURATED ORGANIC COMPOUND NIT2, NOS1, CHRM1 ALDH1A1 948/4885TAAR1 46/4885CYP1A2 212/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.