SCHEMBL9230745

SCHEMBL9230745

COc1cc(OC)nc(SC(C(=O)N(C)[C@@H](C)C(=O)O)C(C)C)n1

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.36
PPARG P37231 1/20 0.36
KDM4E B2RXH2 2/20 0.35
LMNA P02545 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
ADORA1 P30542 1/20 0.35
ALDH1A1 P00352 2/20 0.35
EDNRB P24530 1/20 0.33
EDNRA P25101 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9083549 0.85 ALDH1A1 (0.32) ADORA3ADORA1ALDH1A1
SCHEMBL9082975 0.83 ALOX5 (0.44) ALOX5PPARGKDM4ELMNAALDH1A1
SCHEMBL13851483 0.83 ALOX5 (0.44) ALOX5PPARGKDM4ELMNAALDH1A1
SCHEMBL13851482 0.83 ALOX5 (0.44) ALOX5PPARGKDM4ELMNAALDH1A1
SCHEMBL16160330 0.78 CYP1A2 (0.44) KDM4ELMNAADORA3ADORA1ALDH1A1
SCHEMBL9388237 0.78 ADORA3 (0.41) ALOX5PPARGADORA3ADORA1ALDH1A1
SCHEMBL9401416 0.76 CYP1A2 (0.42) KDM4EADORA3ADORA1ALDH1A1
SCHEMBL9388253 0.76 LMNA (0.38) KDM4ELMNAADORA3ADORA1ALDH1A1
SCHEMBL9082706 0.75 KDM4E (0.39) ALOX5PPARGKDM4ELMNAADORA3
SCHEMBL9084366 0.75 EDNRB (0.44) LMNAEDNRBEDNRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0601155-A1 PYRIMIDINYL-AND TRIAZINYL COMPOUNDS WITH HERBICIDAL ACTIVITY Novartis AG (CH) 1994-06-15 EP claimed
WO-1993025540-A1 PYRIMIDINYL-AND TRIAZINYL COMPOUNDS WITH HERBICIDAL ACTIVITY CIBA-GEIGY AG (CH) 1993-12-23 WO claimed
US-5482920-A Triazinyl compounds with herbicidal activity CIBA-GEIGY CORPORATION (US) 1996-01-09 US disclosed
EP-0601155-A1 PYRIMIDINYL-AND TRIAZINYL COMPOUNDS WITH HERBICIDAL ACTIVITY Novartis AG (CH) 1994-06-15 EP disclosed
WO-1993025540-A1 PYRIMIDINYL-AND TRIAZINYL COMPOUNDS WITH HERBICIDAL ACTIVITY CIBA-GEIGY AG (CH) 1993-12-23 WO disclosed