SCHEMBL9252290

SCHEMBL9252290

CC(=O)N1CCC(CC(=O)c2ccc(N(C)C)cc2)CC1

nearest known ligand 0.67

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.46
DRD2 P14416 2/20 0.46
HTR2A P28223 2/20 0.46
HTR2C P28335 2/20 0.46
HTR2B P41595 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9249556 0.86 BCHE (0.46) DRD2
SCHEMBL11101318 0.84 SIGMAR1 (0.49) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL9253569 0.83 DRD2 (0.66) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL8119451 0.83 CASP6 (0.49) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL11096282 0.83 ALDH1A1 (0.59) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL11095799 0.83 ALDH1A1 (0.55) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL9247360 0.81 CCR5 (0.49) HTR2B
SCHEMBL11095969 0.81 POLB (0.50)
SCHEMBL9255015 0.80 MBTD1 (0.46) SIGMAR1DRD2HTR2AHTR2CHTR2B
SCHEMBL9253376 0.78 HDAC1 (0.45) SIGMAR1DRD2HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5441967-A Treating cerebral edema; anticholinesterase or brain function-improving agent TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-08-15 US disclosed
US-5294625-A 1-benzyl,4-((4-dialkylaminophenyl)carbonyl)piperidines TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-03-15 US disclosed
EP-0378207-B1 CYCLIC AMINE COMPOUNDS AND THEIR USE Takeda Chemical Industries, Ltd. (JP) 1993-09-22 EP disclosed
US-5177087-A Cerebral edema, cholinesterase inhibitor TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-01-05 US disclosed
EP-0378207-A1 Cyclic amine compounds and their use Takeda Chemical Industries, Ltd. (JP) 1990-07-18 EP disclosed