SCHEMBL9254355

SCHEMBL9254355

CC(C)(C)C(=O)OCOC(=O)CCc1cn(-c2ccc(-c3ccc(C(=N)NC(=O)OCc4ccccc4)cc3)nn2)cn1

nearest known ligand 0.35

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 2/20 0.35
MASP2 O00187 2/20 0.31
NPC1 O15118 1/20 0.30
CASP1 P29466 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9257621 0.84 PDK1 (0.36) PDK1MASP2
SCHEMBL9257250 0.83 PDK1 (0.31) PDK1NPC1
SCHEMBL9255067 0.82 PDK1 (0.33) PDK1NPC1
SCHEMBL9250749 0.81 ALOX5 (0.30) PDK1
SCHEMBL9259482 0.80 PDK1 (0.33) PDK1NPC1
SCHEMBL9255100 0.77 KDM4E (0.36) MASP2CASP1
SCHEMBL9260202 0.76 SMN1; SMN2 (0.39) MASP2NPC1CASP1
SCHEMBL9251800 0.73 PDK1 (0.36) PDK1NPC1
SCHEMBL8863938 0.72 TMPRSS15 (0.36) PDK1NPC1
SCHEMBL9568201 0.71 MAPT (0.39) MASP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5463071-A Tetrazole derivatives; useful for inhibiting undesirable cell aggregation DR. KARL THOMAE GMBH (DE) 1995-10-31 US disclosed
EP-0525629-A2 5-membered heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-02-03 EP disclosed