SCHEMBL9257250

SCHEMBL9257250

CC(C)(C)C(=O)OCOC(=O)CCc1cn(-c2ccc(-c3ccc(C(=N)N)cc3)nn2)cn1

nearest known ligand 0.32

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9254094 0.88 F2 (0.37) PDK1NPC1RAB9A
SCHEMBL8863938 0.86 TMPRSS15 (0.36) PDK1NPC1RAB9A
SCHEMBL9257803 0.86 MAPT (0.35)
SCHEMBL9254355 0.83 PDK1 (0.35) PDK1NPC1
SCHEMBL9568440 0.82 ITGB3 (0.39) PDK1
SCHEMBL9250531 0.82 F2 (0.35) PDK1
SCHEMBL9251525 0.81 MIF (0.37) PDK1NPC1
SCHEMBL9254692 0.80 F10 (0.34) PDK1
SCHEMBL9253978 0.79 ITGB3 (0.37) PDK1
SCHEMBL9255067 0.77 PDK1 (0.33) PDK1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5463071-A Tetrazole derivatives; useful for inhibiting undesirable cell aggregation DR. KARL THOMAE GMBH (DE) 1995-10-31 US disclosed
EP-0525629-A2 5-membered heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-02-03 EP disclosed