SCHEMBL9257912

SCHEMBL9257912

N=C(N)c1ccc(-c2ccc(-c3nnc(CCC(=O)O)o3)cc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 1/20 0.61
RAB9A P51151 4/20 0.49
KMT2A Q03164 3/20 0.49
NPC1 O15118 3/20 0.49
MEN1 O00255 2/20 0.49
ALDH1A1 P00352 2/20 0.49
KDM4E B2RXH2 1/20 0.49
PKM P14618 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.46
MAPT P10636 1/20 0.45
HCAR2 Q8TDS4 1/20 0.45
PRSS1 P07477 1/20 0.44
TMPRSS15 P98073 1/20 0.44
NQO2 P16083 1/20 0.43
ITGB3 P05106 1/20 0.43
ITGA2B P08514 1/20 0.43
HDAC3 O15379 1/20 0.43
HDAC4 P56524 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC7 Q8WUI4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9257683 0.85 ITGB3 (0.56) NR1H4RAB9ANPC1MAPTPRSS1
SCHEMBL9250754 0.85 KMT2A (0.49) NR1H4RAB9AKMT2ANPC1MEN1
SCHEMBL561946 0.80 NR1H4 (0.69) NR1H4RAB9AKMT2ANPC1MEN1
SCHEMBL24073125 0.79 NR1H4 (0.64) NR1H4RAB9AKMT2ANPC1MEN1
SCHEMBL9259668 0.78 RXRA (0.71) RAB9ANPC1ALDH1A1KDM4EPRSS1
SCHEMBL17384053 0.74 WDR5 (0.66) RAB9AKMT2ANPC1MEN1ALDH1A1
SCHEMBL3518708 0.73 NR1H4 (0.60) NR1H4RAB9AKMT2ANPC1MEN1
SCHEMBL9254121 0.73 ALDH1A1 (0.64) ALDH1A1KDM4EPKMMAPTPRSS1
Hydrochloric Acid SCHEMBL17377346 0.72 WDR5 (0.63) RAB9AKMT2ANPC1MEN1ALDH1A1
SCHEMBL9255174 0.71 NQO2 (0.67) ALDH1A1PRSS1TMPRSS15NQO2ITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5463071-A Tetrazole derivatives; useful for inhibiting undesirable cell aggregation DR. KARL THOMAE GMBH (DE) 1995-10-31 US disclosed
EP-0525629-A2 5-membered heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-02-03 EP disclosed