SCHEMBL9258798

SCHEMBL9258798

COP(C)(=O)OCC(=O)c1ccc(F)c(F)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.43
CES1 P23141 2/20 0.43
CHRNA1 P02708 1/20 0.38
CHRNG P07510 1/20 0.38
CHRNB1 P11230 1/20 0.38
CHRNB2 P17787 1/20 0.38
SLC6A2 P23975 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA4 P43681 1/20 0.38
SLC6A3 Q01959 1/20 0.38
CHRND Q07001 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
VNN1 O95497 1/20 0.38
TDP1 Q9NUW8 1/20 0.37
RAB9A P51151 2/20 0.37
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9250126 0.83 NPC1 (0.44) MEN1KMT2ARAB9ALMNAMAPK1
SCHEMBL9254905 0.81 NPC1 (0.46) CES2CES1ALDH1A1MEN1KMT2A
SCHEMBL31114440 0.79 CES2 (0.53) CES2CES1CHRNA1CHRNGCHRNB1
SCHEMBL9255947 0.78 NPC1 (0.47) ALDH1A1MEN1KMT2ATDP1RAB9A
SCHEMBL10878397 0.76 POLB (0.57) CES1ALDH1A1MEN1KMT2ATDP1
SCHEMBL9254114 0.76 THRB (0.40) CES2CES1MEN1KMT2ATDP1
SCHEMBL9254524 0.75 CASP3 (0.48) CES2CES1ALDH1A1MEN1KMT2A
SCHEMBL9254186 0.72 GSK3B (0.50) CES1ALDH1A1MEN1KMT2ATDP1
SCHEMBL11548835 0.72 TRPA1 (0.45) ALDH1A1MEN1KMT2ATDP1RAB9A
SCHEMBL25193546 0.71 MEN1 (0.54) CES2CES1CHRNA1CHRNGCHRNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5401768-A Prostaglandin derivative, antiulcer, hypotensive, anticoagulant TORAY INDUSTRIES, INC. (JP) 1995-03-28 US disclosed
EP-0365678-B1 2,5,6,7-TETRANOR-4,8-INTER-m-PHENYLENE PGI 2 DERIVATIVES, PROCESS FOR THEIR PREPARATION, AND USE THEREOF TORAY INDUSTRIES (JP) 1994-01-05 EP disclosed
EP-0365678-A1 2,5,6,7-TETRANOR-4,8-INTER-m-PHENYLENE PGI 2 DERIVATIVES, PROCESS FOR THEIR PREPARATION, AND USE THEREOF TORAY INDUSTRIES, INC. (JP) 1990-05-02 EP disclosed