SCHEMBL9293371

SCHEMBL9293371

C[SiH](C)Oc1c(Br)cc(C(C)(C)C)cc1-c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.34
MAPK1 P28482 1/20 0.34
BACE1 P56817 1/20 0.32
NPC1 O15118 1/20 0.32
PLA2G1B P04054 1/20 0.32
NFKB1 P19838 1/20 0.32
CASP3 P42574 1/20 0.32
RAB9A P51151 1/20 0.32
NFKB2 Q00653 1/20 0.32
RELA Q04206 1/20 0.32
SENP8 Q96LD8 1/20 0.32
SENP7 Q9BQF6 1/20 0.32
SENP6 Q9GZR1 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
ATG4B Q9Y4P1 1/20 0.32
RXRA P19793 3/20 0.31
RXRB P28702 3/20 0.31
PDE4A P27815 1/20 0.31
PDE4B Q07343 1/20 0.31
PDE4C Q08493 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3415618 0.83 PDE4B (0.43) ALDH1A1MAPK1BACE1NPC1PLA2G1B
SCHEMBL9293119 0.77 AKR1C3 (0.36) NPC1RAB9A
SCHEMBL13376117 0.77 EGFR (0.38) ALDH1A1MAPK1PDE4APDE4BPDE4C
SCHEMBL13508914 0.77 THRB (0.44) ALDH1A1MEN1KMT2A
SCHEMBL13044012 0.76 THRA (0.42) MAPK1RXRARXRBRXRG
SCHEMBL9293194 0.75 KIF11 (0.40) ALDH1A1MAPK1NPC1PLA2G1BNFKB1
SCHEMBL13773460 0.74 PDE4B (0.49) ALDH1A1BACE1NPC1PLA2G1BNFKB1
SCHEMBL3418407 0.73 CRHBP (0.48) ALDH1A1MAPK1BACE1NPC1PLA2G1B
SCHEMBL25976215 0.73 NPC1 (0.38) ALDH1A1MAPK1BACE1NPC1PLA2G1B
Potassium Ion SCHEMBL3416456 0.72 ALDH1A1 (0.38) ALDH1A1MAPK1BACE1NPC1PLA2G1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5350846-A Antibiotics MERCK & CO., INC. (US) 1994-09-27 US disclosed
US-5208329-A Antibacterial agents MERCK & CO., INC. (US) 1993-05-04 US disclosed
US-5182385-A Chemical intermediates for bactericides MERCK & CO., INC. (US) 1993-01-26 US disclosed
EP-0467434-A1 2-Biphenyl-carbapenem antibacterial agents MERCK & CO. INC. (US) 1992-01-22 EP disclosed
EP-0464900-A2 2-Biphenyl-carbapenems MERCK & CO. INC. (US) 1992-01-08 EP disclosed
US-5025006-A Carbapenicillin antibiotics MERCK & CO., INC. (US) 1991-06-18 US disclosed
US-5011832-A 2-biphenyl-carbapenem antibacterial agents MERCK & CO., INC. (US) 1991-04-30 US disclosed