SCHEMBL9303445

SCHEMBL9303445

N=C(N)Nc1ccccc1C(=O)Nc1cccc2c(C(=N)N)cccc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.54
RAB9A P51151 3/20 0.54
KDM4E B2RXH2 3/20 0.50
SMN1; SMN2 Q16637 3/20 0.50
POLB P06746 1/20 0.50
PARP1 P09874 2/20 0.48
CHRNB2 P17787 1/20 0.48
CHRNB4 P30926 1/20 0.48
CHRNA3 P32297 1/20 0.48
CHRNA4 P43681 1/20 0.48
GAA P10253 3/20 0.47
ALDH1A1 P00352 4/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
TP53 P04637 1/20 0.47
NFKB1 P19838 1/20 0.47
NFKB2 Q00653 1/20 0.47
RELA Q04206 1/20 0.47
MAPT P10636 1/20 0.46
PPARG P37231 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9303104 0.96 NPC1 (0.49) NPC1RAB9AKDM4ESMN1; SMN2POLB
SCHEMBL9302237 0.88 F10 (0.49) NPC1RAB9AKDM4ESMN1; SMN2POLB
SCHEMBL9303405 0.82 NPC1 (0.48) NPC1RAB9AKMT2ACYP1A2CYP3A4
SCHEMBL9302810 0.82 NPC1 (0.49) NPC1RAB9AKDM4ESMN1; SMN2POLB
SCHEMBL9303484 0.81 NPC1 (0.49) NPC1RAB9AKDM4ESMN1; SMN2POLB
SCHEMBL9303308 0.80 PTGES (0.56) NPC1RAB9AGAAMEN1KMT2A
SCHEMBL9302799 0.80 RXFP1 (0.50) NPC1RAB9AKDM4ESMN1; SMN2POLB
SCHEMBL9303274 0.80 PLAU (0.62) NPC1RAB9AKDM4ESMN1; SMN2POLB
SCHEMBL9303507 0.80 KDM4E (0.47) NPC1RAB9AKDM4ESMN1; SMN2POLB
SCHEMBL9302926 0.80 RAB9A (0.50) NPC1RAB9AKDM4ESMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5352704-A Antiviral agents BANYU PHARMACEUTICAL CO., LTD. (JP) 1994-10-04 US disclosed
EP-0434432-B1 Guanidinobenzene derivatives BANYU PHARMA CO LTD (JP) 1994-05-04 EP disclosed
EP-0434432-A1 Guanidinobenzene derivatives BANYU PHARMACEUTICAL CO., LTD. (JP) 1991-06-26 EP disclosed