SCHEMBL9305370

SCHEMBL9305370

Sc1nc2cccc(Br)c2[nH]1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 1/20 0.41
CA12 O43570 1/20 0.40
CA9 Q16790 1/20 0.40
DYRK1A Q13627 4/20 0.39
CDK9 P50750 3/20 0.39
DYRK1B Q9Y463 3/20 0.39
DYRK2 Q92630 2/20 0.39
BACE1 P56817 1/20 0.36
PDPK1 O15530 1/20 0.35
GUSB P08236 1/20 0.33
TYMS P04818 1/20 0.31
PDGFRB P09619 1/20 0.30
FGFR1 P11362 1/20 0.30
FGFR3 P22607 1/20 0.30
C1R P00736 1/20 0.30
KMT2A Q03164 1/20 0.30
NISCH Q9Y2I1 1/20 0.30
ENPP3 O14638 1/20 0.30
ENPP1 P22413 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28412208 0.79 PSMD14 (0.33)
SCHEMBL248855 0.79 NOS1 (0.44) NOS1CA12CA9DYRK1ACDK9
SCHEMBL9306986 0.76 ACHE (0.43) GUSBKMT2A
SCHEMBL20479323 0.76 PDPK1 (0.43) NOS1CA12CA9DYRK1ACDK9
SCHEMBL110725 0.76 ALDH1A1 (0.41)
SCHEMBL9306736 0.76 CA12 (0.40) CA12CA9DYRK1ATYMS
SCHEMBL9187598 0.76 MAPT (0.37) TYMSKMT2A
SCHEMBL9502126 0.76 PARP1 (0.44) NOS1CA12CA9DYRK1ACDK9
SCHEMBL18340923 0.76 MASP2 (0.48) NOS1CA12CA9DYRK1ACDK9
SCHEMBL17821369 0.76 NOS1 (0.41) NOS1CA12CA9DYRK1ACDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5347008-A Thio(cyclo) alkanepolycarboxylic acids containing heterocyclic substituents CIBA-GEIGY CORPORATION (US) 1994-09-13 US disclosed
EP-0129506-A2 Heterocyclically substituted thio(cyclo)alkane polycarboxylic acids CIBA-GEIGY AG (CH) 1984-12-27 EP disclosed