SCHEMBL9306986

SCHEMBL9306986

Oc1cccc2nc(S)[nH]c12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.43
ALDH1A1 P00352 2/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
AURKA O14965 2/20 0.37
GUSB P08236 3/20 0.37
KDM4E B2RXH2 2/20 0.37
HPGD P15428 2/20 0.37
F7 P08709 1/20 0.36
PSMB8 P28062 1/20 0.35
CYP1A2 P05177 3/20 0.35
PARP1 P09874 3/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
NQO2 P16083 1/20 0.34
TNKS O95271 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28412208 0.79 PSMD14 (0.33) ALDH1A1MAPTRAB9ANPSR1KDM4E
SCHEMBL4314005 0.79 ACHE (0.46) ACHEALDH1A1GAAMAPTRAB9A
Bromide SCHEMBL11628989 0.78 ACHE (0.45) ACHEALDH1A1GAAMAPTRAB9A
SCHEMBL9187598 0.76 MAPT (0.37) ALDH1A1GAAMAPTRAB9AKMT2A
SCHEMBL110725 0.76 ALDH1A1 (0.41) ALDH1A1GAAMAPTRAB9ANPSR1
SCHEMBL9305473 0.76 ACHE (0.43) ACHEALDH1A1GAAMAPTRAB9A
SCHEMBL9306736 0.76 CA12 (0.40) ALDH1A1MAPTRAB9AKDM4EHPGD
SCHEMBL9305370 0.76 NOS1 (0.41) KMT2AGUSB
SCHEMBL21708401 0.76 ALDH1A1 (0.48) ACHEALDH1A1GAAMAPTRAB9A
SCHEMBL4612577 0.76 PARP1 (0.50) ACHEALDH1A1GAAMAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5347008-A Thio(cyclo) alkanepolycarboxylic acids containing heterocyclic substituents CIBA-GEIGY CORPORATION (US) 1994-09-13 US disclosed
EP-0161220-B1 PROCESS FOR THE PREPARATION OF BETA-(BENZOTHIAZOLYLTHIO) AND BETA (BENZIMIDAZOLYLTHIO)CARBOXYLIC-ACID DERIVATIVES CIBA-GEIGY AG (CH) 1991-08-14 EP disclosed
US-4612378-A Process for the preparation of β-(benzothiazolylthio)- and β-(benzimidazolylthio-carboxylic acids CIBA-GEIGY CORPORATION (US) 1986-09-16 US disclosed
EP-0161220-A2 Process for the preparation of beta-(benzothiazolylthio) and beta (benzimidazolylthio)carboxylic-acid derivatives CIBA-GEIGY AG (CH) 1985-11-13 EP disclosed
EP-0129506-A2 Heterocyclically substituted thio(cyclo)alkane polycarboxylic acids CIBA-GEIGY AG (CH) 1984-12-27 EP disclosed
EP-0126030-A2 Process for the preparation of beta-(benzothiazolylthio) and beta-(benzimidazolylthio) carboxylic acids CIBA-GEIGY AG (CH) 1984-11-21 EP disclosed