SCHEMBL9307022

SCHEMBL9307022

O=C(Nc1ccccc1)c1ccc2sc(S)nc2c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.57
NPC1 O15118 3/20 0.57
ALDH1A1 P00352 3/20 0.57
LMNA P02545 1/20 0.57
MAPT P10636 3/20 0.57
POLB P06746 2/20 0.57
HPGD P15428 2/20 0.57
HDAC1 Q13547 2/20 0.55
SMN1; SMN2 Q16637 2/20 0.51
PKM P14618 1/20 0.51
NFKB1 P19838 1/20 0.51
NFKB2 Q00653 1/20 0.51
RELA Q04206 1/20 0.51
HTT P42858 2/20 0.50
PLAU P00749 2/20 0.49
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
KDM4E B2RXH2 1/20 0.48
USP2 O75604 1/20 0.48
ALOX15 P16050 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9734141 0.80 THRB (0.56) RAB9ANPC1HDAC1SMN1; SMN2PLAU
SCHEMBL2031602 0.79 NPC1 (0.68) RAB9ANPC1ALDH1A1LMNAMAPT
SCHEMBL9306708 0.75 NPC1 (0.49) RAB9ANPC1ALDH1A1HPGDHDAC1
SCHEMBL9305296 0.74 PIK3CA (0.50) RAB9ANPC1ALDH1A1LMNAMAPT
SCHEMBL24124689 0.74 RAB9A (0.56) RAB9ANPC1ALDH1A1LMNAMAPT
SCHEMBL24124970 0.74 GPR27 (0.62) RAB9ANPC1ALDH1A1LMNAMAPT
SCHEMBL7452674 0.73 RAB9A (0.65) RAB9ANPC1ALDH1A1LMNAMAPT
SCHEMBL9305825 0.73 NPC1 (0.72) RAB9ANPC1ALDH1A1LMNAMAPT
SCHEMBL24124852 0.73 RAB9A (0.54) RAB9ANPC1ALDH1A1LMNAMAPT
SCHEMBL9734495 0.73 SMN1; SMN2 (0.52) RAB9ANPC1ALDH1A1MAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5347008-A Thio(cyclo) alkanepolycarboxylic acids containing heterocyclic substituents CIBA-GEIGY CORPORATION (US) 1994-09-13 US disclosed
US-5152929-A Corrosion inhibitors for water systems CIBA-GEIGY CORPORATION (US) 1992-10-06 US disclosed
EP-0129506-B1 HETEROCYCLICALLY SUBSTITUTED THIO(CYCLO)ALKANE POLYCARBOXYLIC ACIDS CIBA-GEIGY AG (CH) 1991-03-06 EP disclosed
US-4652653-A Process for the preparation of β-(benzothiazolylthio)- and β-(benzimidazolylthio)-carboxylic acid derivatives CIBA-GEIGY CORPORATION (US) 1987-03-24 US disclosed
US-4612378-A Process for the preparation of β-(benzothiazolylthio)- and β-(benzimidazolylthio-carboxylic acids CIBA-GEIGY CORPORATION (US) 1986-09-16 US disclosed
EP-0161220-A2 Process for the preparation of beta-(benzothiazolylthio) and beta (benzimidazolylthio)carboxylic-acid derivatives CIBA-GEIGY AG (CH) 1985-11-13 EP disclosed
EP-0129506-A2 Heterocyclically substituted thio(cyclo)alkane polycarboxylic acids CIBA-GEIGY AG (CH) 1984-12-27 EP disclosed
EP-0126030-A2 Process for the preparation of beta-(benzothiazolylthio) and beta-(benzimidazolylthio) carboxylic acids CIBA-GEIGY AG (CH) 1984-11-21 EP disclosed