SCHEMBL932927

SCHEMBL932927

Nc1ccc(COC(=O)OCc2ccc(N)cc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.45
MEN1 O00255 1/20 0.45
ALDH1A1 P00352 4/20 0.44
CYP3A4 P08684 2/20 0.44
TDP1 Q9NUW8 2/20 0.44
GFER P55789 1/20 0.44
TSHR P16473 1/20 0.44
MAOA P21397 2/20 0.44
LMNA P02545 1/20 0.44
CYP1A2 P05177 1/20 0.44
MAOB P27338 3/20 0.42
APP P05067 1/20 0.42
LOXL2 Q9Y4K0 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.41
RAB9A P51151 2/20 0.41
MAPK1 P28482 1/20 0.41
SLC6A2 P23975 1/20 0.41
SLC6A3 Q01959 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27400293 0.92 ALDH1A1 (0.55) KMT2AALDH1A1TDP1MAOALMNA
SCHEMBL29026626 0.88 PPID (0.43) KMT2AMEN1ALDH1A1CYP3A4TSHR
SCHEMBL147245 0.84 KMT2A (0.44) KMT2AMEN1ALDH1A1CYP3A4TDP1
SCHEMBL25448604 0.84 KMT2A (0.44) KMT2AMEN1ALDH1A1CYP3A4TDP1
SCHEMBL1561073 0.84 ALDH1A1 (0.45) KMT2AMEN1ALDH1A1CYP3A4TDP1
SCHEMBL6453211 0.83 ALDH1A1 (0.47) KMT2AMEN1ALDH1A1CYP3A4TDP1
SCHEMBL2511445 0.83 ALDH1A1 (0.64) KMT2AMEN1ALDH1A1CYP3A4TDP1
SCHEMBL27353978 0.83 APP (0.44) KMT2AMEN1ALDH1A1CYP3A4TDP1
SCHEMBL4509522 0.83 ALDH1A1 (0.64) KMT2AMEN1ALDH1A1CYP3A4TDP1
SCHEMBL28625515 0.82 KMT2A (0.52) KMT2AMEN1ALDH1A1CYP3A4TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 85 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260125418-A1 A COMPOUND AND ITS USE FOR DETECTING A DISEASE IN THE EXHALED BREATH OF A SUBJECT OWLSTONE MED LTD (GB) 2026-05-07 US claimed
EP-4598592-A1 A COMPOUND AND ITS USE FOR DETECTING A DISEASE IN THE EXHALED BREATH OF A SUBJECT Owlstone Medical Limited (GB) 2025-08-13 EP claimed
CN-120152745-A Compounds and their use for detecting diseases in exhaled breath of a subject 奥斯通医疗有限公司 2025-06-13 CN claimed
WO-2025031383-A1 BIFUNCTIONAL LINKER COMPOUND, ANTIBODY DRUG CONJUGATE, PREPARATION METHOD FOR ANTIBODY DRUG CONJUGATE, AND USE OF ANTIBODY DRUG CONJUGATE 杭州爱科瑞思生物医药有限公司 2025-02-13 WO claimed
WO-2024074813-A1 A COMPOUND AND ITS USE FOR DETECTING A DISEASE IN THE EXHALED BREATH OF A SUBJECT OWLSTONE MEDICAL LIMITED (GB) 2024-04-11 WO claimed
CN-117069793-A Bifunctional linker compound, antibody drug conjugate, and preparation methods and applications thereof 杭州爱科瑞思生物医药有限公司 2023-11-17 CN claimed
EP-4079316-A1 PROCOAGULANT COMPOUNDS Bioverativ Therapeutics Inc. (US) 2022-10-26 EP claimed
US-20220243189-A1 PROCOAGULANT COMPOUNDS BIOGEN MA INC. 2022-08-04 US claimed
EP-3693000-B1 PROCOAGULANT COMPOUNDS BIOVERATIV THERAPEUTICS INC (US) 2022-03-02 EP claimed
EP-3693000-A1 PROCOAGULANT COMPOUNDS Bioverativ Therapeutics Inc. (US) 2020-08-12 EP claimed
WO-2015187540-A1 PEPTIDE-DRUG CONJUGATES CHU SHAOSONG (US) 2015-12-10 WO claimed
US-20150343083-A1 PEPTIDE-DRUG CONJUGATES JIARAY PHARMACEUTICALS, INC. (KY) 2015-12-03 US claimed
US-20150328330-A1 CONJUGATES OF A POLYMER, A BISPHOSPHONATE AND AN ANTI-ANGIOGENESIS AGENT AND USES THEREOF IN THE TREATMENT AND MONITORING OF BONE RELATED DISEASES RAMOT AT TEL-AVIV UNIVERSITY LTD. (IL) 2015-11-19 US claimed
US-9095618-B2 Conjugates of a polymer, a bisphosphonate and an anti-angiogenesis agent and uses thereof in the treatment and monitoring of bone related diseases RAMOT AT TEL-AVIV UNIVERSITY LTD. (IL) 2015-08-04 US claimed
US-20150184142-A1 PROCOAGULANT COMPOUNDS BIOGEN IDEC MA INC. (US) 2015-07-02 US claimed
US-20140134111-A1 CONJUGATES OF A POLYMER, A BISPHOSPHONATE AND AN ANTI-ANGIOGENESIS AGENT AND USES THEREOF IN THE TREATMENT AND MONITORING OF BONE RELATED DISEASES RAMOT AT TEL-AVIV UNIVERSITY LTD. (IL) 2014-05-15 US claimed
US-8658149-B2 Conjugates of a polymer, a bisphosphonate and an anti-angiogenesis agent and uses thereof in the treatment and monitoring of bone related diseases RAMOT AT TEL-AVIV UNIVERSITY LTD. (IL) 2014-02-25 US claimed
US-20110142764-A1 CONJUGATES OF A POLYMER, A BISPHOSPHONATE AND AN ANTI-ANGIOGENESIS AGENT AND USES THEREOF IN THE TREATMENT AND MONITORING OF BONE RELATED DISEASES RAMOT AT TEL-AVIV UNIVERSITY LTD. (IL) 2011-06-16 US claimed
EP-2303288-A2 CONJUGATES OF A POLYMER, A BISPHOSPHONATE AND AN ANTI-ANGIOGENESIS AGENT AND USES THEREOF IN THE TREATMENT AND MONITORING OF BONE RELATED DISEASES Ramot at Tel-Aviv University Ltd. (IL) 2011-04-06 EP claimed
WO-2009141823-A2 CONJUGATES OF A POLYMER, A BISPHOSPHONATE AND AN ANTI-ANGIOGENESIS AGENT AND USES THEREOF IN THE TREATMENT AND MONITORING OF BONE RELATED DISEASES RAMOT AT TEL AVIV UNIVERSITY LTD. (IL) 2009-11-26 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150328330-A1 CONJUGATES OF A POLYMER, A BISPHOSPHONATE AND AN ANTI-ANGIOGENESIS AGENT AND USES THEREOF IN THE TREATMENT AND MONITORING OF BONE RELATED DISEASES VEGFA, BPGM, SOST KMT2A 4124/4885MEN1 1384/4885ALDH1A1 2685/4885
US-20260125418-A1 A COMPOUND AND ITS USE FOR DETECTING A DISEASE IN THE EXHALED BREATH OF A SUBJECT BRCA1, L3MBTL1, LMNA KMT2A 3488/4885MEN1 35/4885ALDH1A1 1039/4885
US-20220243189-A1 PROCOAGULANT COMPOUNDS PLG, F2, PLAT KMT2A 3722/4885MEN1 1483/4885ALDH1A1 4124/4885
US-20150184142-A1 PROCOAGULANT COMPOUNDS PLG, F2, PLAT KMT2A 3722/4885MEN1 1483/4885ALDH1A1 4124/4885
US-20150343083-A1 PEPTIDE-DRUG CONJUGATES DNPEP, VIP, PEPD KMT2A 3657/4885MEN1 482/4885ALDH1A1 3736/4885
US-20140134111-A1 CONJUGATES OF A POLYMER, A BISPHOSPHONATE AND AN ANTI-ANGIOGENESIS AGENT AND USES THEREOF IN THE TREATMENT AND MONITORING OF BONE RELATED DISEASES VEGFA, BPGM, SOST KMT2A 4124/4885MEN1 1384/4885ALDH1A1 2685/4885
US-20110142764-A1 CONJUGATES OF A POLYMER, A BISPHOSPHONATE AND AN ANTI-ANGIOGENESIS AGENT AND USES THEREOF IN THE TREATMENT AND MONITORING OF BONE RELATED DISEASES VEGFA, BPGM, SOST KMT2A 4124/4885MEN1 1384/4885ALDH1A1 2685/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.