Water

Water

SCHEMBL93584

Cc1ccccc1C(C)(C)N.O

nearest known ligand 0.43

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Water. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE known ✓ P22303 2/20 0.43
SLC6A2 known ✓ P23975 1/20 0.34
TSHR P16473 3/20 0.43
GABRA1 P14867 1/20 0.41
GABRB2 P47870 1/20 0.41
CASR P41180 1/20 0.40
TDP1 Q9NUW8 2/20 0.39
CYP3A4 P08684 1/20 0.39
ALDH1A1 P00352 3/20 0.36
CA2 P00918 2/20 0.35
CA1 P00915 1/20 0.35
CA7 P43166 1/20 0.35
CA9 Q16790 1/20 0.35
TAAR1 Q96RJ0 2/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
CYP2A6 P11509 2/20 0.32
CD44 P16070 1/20 0.32
TRPA1 O75762 1/20 0.32
ATM Q13315 1/20 0.32
CYP1A2 P05177 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL164361 0.97 TSHR (0.45) TSHRACHEGABRA1GABRB2CASR
SCHEMBL29581427 0.97 TSHR (0.45) TSHRACHEGABRA1GABRB2CASR
Methyl Alcohol SCHEMBL5165690 0.95 GABRA1 (0.43) TSHRACHEGABRA1GABRB2CASR
Iodide SCHEMBL1502892 0.95 TSHR (0.43) TSHRACHEGABRA1GABRB2CASR
Bromide SCHEMBL21460045 0.95 TSHR (0.43) TSHRACHEGABRA1GABRB2CASR
Hydrochloric Acid SCHEMBL23886258 0.95 TDP1 (0.44) TSHRACHEGABRA1GABRB2CASR
Fluoride SCHEMBL1502827 0.95 TSHR (0.43) TSHRACHEGABRA1GABRB2CASR
Bromide SCHEMBL622796 0.95 TSHR (0.43) TSHRACHEGABRA1GABRB2CASR
Ammonia Solution, Strong SCHEMBL5145133 0.95 TSHR (0.43) TSHRACHEGABRA1GABRB2CASR
Hydrochloric Acid SCHEMBL136350 0.95 TDP1 (0.44) TSHRACHEGABRA1GABRB2CASR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 3405 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4605578-A2 ELECTROCATALYTIC GENERATION OF IMINES FROM ALCOHOLS AND AMINES Université Paris Cité (FR) 2025-08-27 EP claimed
WO-2025102202-A1 POLYISOCYANATE COMPOSITION, AND COATING LAYER HAVING IMPROVED CHEMICAL RESISTANCE 万华化学集团股份有限公司 2025-05-22 WO claimed
CN-119978314-A Polyisocyanate composition and coating with improved chemical resistance 万华化学集团股份有限公司 2025-05-13 CN claimed
CN-119798515-A Hydrogel-based super stretch-proof flexible multifunctional input device and preparation and application thereof 北京大学 2025-04-11 CN claimed
CN-114685378-B Preparation method of 4, 6-dihydroxypyrimidine 南通泰禾化工股份有限公司 2025-03-04 CN claimed
CN-119144236-A Polishing solution and preparation method thereof 江苏山水半导体科技有限公司 2024-12-17 CN claimed
EP-4470056-A1 NOVEL AQUEOUS-PHASE REDOX FLOW BATTERIES Kemiwatt (FR) 2024-12-04 EP claimed
CN-118493978-B Waterproof breathable polyester fiber fabric and production process thereof 安徽金弘润新材料科技有限公司 2024-09-10 CN claimed
CN-118493978-A Waterproof breathable polyester fiber fabric and production process thereof 安徽金弘润新材料科技有限公司 2024-08-16 CN claimed
CN-117700710-B Phosphorus-containing polycarbonate resin and preparation method and application thereof 拓烯科技(衢州)有限公司 2024-08-09 CN claimed
EP-0524501-B1 A process for the production of polyisocyanates containing allophanate and isocyanurate groups BAYER AG (US) 1996-10-30 EP claimed
US-5162452-A Coatings WACKER-CHEMIE GMBH (DE) 1992-11-10 US claimed
US-4730049-A Process for preparing 5-(2-chlorobenzyl)-4,5,6,7-tetrahydrothieno (3,2-C)pyridine NISSHIN FLOUR MILLING CO., LTD. (JP) 1988-03-08 US claimed
US-4726835-A Herbicidal and plant growth regulating imidazoline derivatives IDEMITSU KOSAN COMPANY LIMITED (JP) 1988-02-23 US claimed
US-4584410-A HYDROXIDE OR OXIDE OF ALKALI OR ALKALINE METAL DECOMPOSES CONTAMIN SUMITOMO CHEMICAL CO., LTD. (JP) 1986-04-22 US claimed
US-4443590-A ISOCYANATE COMPONENT HAVING OXADIAZINETRIONE RING, ACTIVE HYDROGEN COMPONENT, LEWIS BASE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1984-04-17 US claimed
US-4214057-A Coating composition for plastic substrates ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1980-07-22 US claimed
US-4192820-A Preparation of 3-methyl-2-buten-1-al BASF AKTIENGESELLSCHAFT (DE) 1980-03-11 US claimed
US-4163757-A ACIDIC CLAY CATALYST THE GOODYEAR TIRE & RUBBER COMPANY (US) 1979-08-07 US claimed
US-4152340-A BY REACTING 1,4,4A,5,8,8A,9A,10A-OCTAHYDRO-ANTHRAQUINONE WITH NITROBENZENE, BASIC COMPOUND, INHIBITOR PRODUITS CHIMIQUES UGINE KUHLMANN (FR) 1979-05-01 US claimed