SCHEMBL9429140

SCHEMBL9429140

CCN(CCNCCOc1ccc(C#N)cc1)c1cc(=O)n(C)c(=O)n1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 1/20 0.37
MMP2 P08253 3/20 0.37
MMP3 P08254 3/20 0.37
DRD2 P14416 1/20 0.36
DRD4 P21917 1/20 0.36
DRD3 P35462 1/20 0.36
CYP19A1 P11511 4/20 0.35
CACNA1B Q00975 2/20 0.35
HRH2 P25021 1/20 0.35
HRH1 P35367 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
CACNA1H O95180 1/20 0.35
ALDH1A1 P00352 3/20 0.35
MAPT P10636 1/20 0.35
TBXAS1 P24557 1/20 0.35
POLB P06746 1/20 0.35
PKM P14618 1/20 0.35
HPGD P15428 1/20 0.35
KCNA5 P22460 1/20 0.35
GFER P55789 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9428502 0.85 DRD2 (0.47) DRD2DRD4DRD3ALDH1A1
SCHEMBL9386345 0.84 DRD2 (0.51) DRD2DRD4DRD3ALDH1A1MAPT
SCHEMBL9385003 0.82 PKM (0.52) DRD2DRD4DRD3HRH2HRH1
SCHEMBL9429147 0.78 SCN8A (0.38) DRD4CYP19A1CACNA1BHRH3POLB
SCHEMBL9428964 0.77 MAPK1 (0.49) RXFP1MMP3DRD2DRD4DRD3
SCHEMBL9428388 0.72 CYP1A2 (0.49) RXFP1MMP3DRD2DRD3HRH1
SCHEMBL9428759 0.71 ADRB2 (0.38) RXFP1ALDH1A1HPGD
SCHEMBL1715002 0.71 MMP3 (0.55) MMP2MMP3DRD2DRD4DRD3
SCHEMBL8780756 0.69 ADORA3 (0.40) RXFP1MMP2MMP3CYP19A1MAPT
SCHEMBL1714696 0.69 DRD4 (0.58) MMP3DRD2DRD4DRD3HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5332739-A Pyrimidinedione derivatives and antiarrhythmic agents containing same MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1994-07-26 US disclosed
EP-0454498-A2 Pyrimidinedione derivatives and antiarrhythmic agents containing same MITSUI TOATSU CHEMICALS, Inc. (JP) 1991-10-30 EP disclosed