SCHEMBL9434693

SCHEMBL9434693

O=C(C=Cc1cccc(Br)c1)Cc1cccnc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.56
CYP2D6 P10635 3/20 0.56
CYP1B1 Q16678 3/20 0.56
CYP3A4 P08684 2/20 0.56
CYP1A1 P04798 2/20 0.56
BACE1 P56817 1/20 0.53
HSD17B3 P37058 1/20 0.52
HDAC4 P56524 1/20 0.49
MEF2D Q14814 1/20 0.49
PLAAT5 Q96KN8 1/20 0.49
PLAAT4 Q9UL19 1/20 0.49
SLC6A19 Q695T7 1/20 0.47
MAPT P10636 2/20 0.47
LMNA P02545 2/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
KMT2A Q03164 1/20 0.47
NAPRT Q6XQN6 1/20 0.47
TBXAS1 P24557 2/20 0.46
IDO1 P14902 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9434748 0.86 CYP1A1 (0.62) CYP1A2CYP1B1CYP1A1HDAC4MEF2D
SCHEMBL9434018 0.85 TBXAS1 (0.56) CYP1A2CYP2D6CYP1B1CYP3A4CYP1A1
SCHEMBL9433864 0.85 NAPRT (0.47) CYP1A2CYP2D6CYP1B1CYP3A4CYP1A1
SCHEMBL9434440 0.85 LMNA (0.47) CYP1A2CYP2D6CYP1B1CYP3A4CYP1A1
SCHEMBL15943749 0.84 HSD17B3 (0.61) CYP2D6CYP1B1BACE1HSD17B3HDAC4
SCHEMBL9434590 0.81 P4HB (0.58) MAPTLMNAKMT2APKMMAOA
SCHEMBL9434552 0.81 P4HB (0.48) HDAC4MEF2DMAPTLMNANAPRT
SCHEMBL9434737 0.81 ALDH1A1 (0.52) CYP1A2CYP2D6CYP1B1CYP3A4CYP1A1
SCHEMBL9433920 0.81 TBXAS1 (0.56) CYP1A2CYP2D6CYP1B1CYP3A4CYP1A1
SCHEMBL7382581 0.81 TGM2 (0.66) MAPTLMNAKDM4ENPC1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5276150-A Vasodilators, anticoagulants, calcium channel blockers FUJIREBIO INC. (JP) 1994-01-04 US disclosed
EP-0400660-A1 1,4-dihydropyridine derivatives FUJIREBIO INC. (JP) 1990-12-05 EP disclosed