Antergan

Antergan

SCHEMBL94485

CN(C)CCN(Cc1ccccc1)c1ccccc1

nearest known ligand 0.66

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.62
CHRM2 P08172 2/20 0.60
ADRA2A P08913 2/20 0.60
DRD1 P21728 2/20 0.60
SLC6A2 P23975 2/20 0.60
SLC6A4 P31645 2/20 0.60
ADRA1A P35348 2/20 0.60
SLC6A3 Q01959 2/20 0.60
KCNH2 Q12809 2/20 0.60
ADRA2B P18089 1/20 0.60
ADRA2C P18825 1/20 0.60
HTR2A P28223 1/20 0.60
HRH1 P35367 1/20 0.60
OPRK1 P41145 1/20 0.60
KDM4E B2RXH2 3/20 0.58
LMNA P02545 3/20 0.58
SMN1; SMN2 Q16637 2/20 0.58
MAPK1 P28482 1/20 0.58
ALDH1A1 P00352 3/20 0.56
CYP2C19 P33261 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7565830 0.88 CHRM2 (0.53) TSHRCHRM2ADRA2ADRD1SLC6A2
SCHEMBL14980578 0.88 TSHR (0.62) TSHRCHRM2ADRA2ADRD1SLC6A2
SCHEMBL11501576 0.85 TAAR1 (0.50) TSHRCHRM2ADRA2ADRD1SLC6A2
SCHEMBL13061113 0.85 TSHR (0.50) TSHRCHRM2ADRA2ADRD1SLC6A2
SCHEMBL13006267 0.84 CHRM2 (0.49) TSHRCHRM2ADRA2ADRD1SLC6A2
SCHEMBL10650495 0.82 TSHR (0.59) TSHRCHRM2ADRA2ADRD1SLC6A2
SCHEMBL641218 0.82 TSHR (0.70) TSHRADRA2AADRA1ASLC6A3KCNH2
SCHEMBL13005467 0.81 ADRA2B (0.47) TSHRCHRM2ADRA2ADRD1SLC6A2
SCHEMBL11174747 0.81 TSHR (0.85) TSHRCHRM2ADRA2ADRD1SLC6A2
SCHEMBL43183 0.80 TSHR (0.74) TSHRADRA2AADRA1ASLC6A3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 358 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1832287-B1 The use of histamine receptor antagonists for the reduction of intracranial pressure JANSSEN PHARMACEUTICA NV (BE) 2009-02-25 EP claimed
EP-1986614-A2 PROTEIN HYDROLYSATE EXCIPIENTS Wyeth (US) 2008-11-05 EP claimed
EP-1165048-A4 COMPOSITIONS AND METHODS FOR IMPROVED DELIVERY OF IONIZABLE HYDROPHOBIC THERAPEUTIC AGENTS LIPOCINE INC (US) 2007-12-05 EP claimed
EP-1832287-A2 The use of anti-histaminics for acute reduction of elevated intracranial pressure JANSSEN PHARMACEUTICA N.V. (BE) 2007-09-12 EP claimed
EP-1829527-A2 Aggregate with increased deformability, comprising at least three amphipats, for improved transport through semi-permeable barriers and for the non-invasive drug application in vivo, especially through the skin IDEA AG (DE) 2007-09-05 EP claimed
EP-1829528-A2 Aggregate with increased deformability, comprising at least three amphipats, for improved transport through semi-permeable barriers and for the non-invasive drug application in vivo, especially through the skin IDEA AG (DE) 2007-09-05 EP claimed
WO-2007097936-A2 PROTEIN HYDROLYSATE EXCIPIENTS WYETH (US) 2007-08-30 WO claimed
US-20070190130-A1 Protein hydrolysate excipients WYETH 2007-08-16 US claimed
EP-1815846-A2 Aggregate with increased deformability, comprising at least three amphipats, for improved transport through semi-permeable barriers and for the non-invasive drug application in vivo, especially through the skin IDEA AG (DE) 2007-08-08 EP claimed
EP-1815847-A2 Aggregate with increased deformability, comprising at least three amphipats, for improved transport through semi-permeable barriers and for the non-invasive drug application in vivo, especially through the skin IDEA AG (DE) 2007-08-08 EP claimed
EP-1551370-A1 AGGREGATE WITH INCREASED DEFORMABILITY, COMPRISING AT LEAST THREE AMPHIPATS, FOR IMPROVED TRANSPORT THROUGH SEMI-PERMEABLE BARRIERS AND FOR THE NON-INVASIVE DRUG APPLICATION IN VIVO, ESPECIALLY THROUGH THE SKIN IDEA AG (DE) 2005-07-13 EP claimed
US-20040105881-A1 Aggregates with increased deformability, comprising at least three amphipats, for improved transport through semi-permeable barriers and for the non-invasive drug application in vivo, especially through the skin IDEA AG (DE) 2004-06-03 US claimed
WO-2004032900-A1 AGGREGATE WITH INCREASED DEFORMABILITY, COMPRISING AT LEAST THREE AMPHIPATS, FOR IMPROVED TRANSPORT THROUGH SEMI-PERMEABLE BARRIERS AND FOR THE NON-INVASIVE DRUG APPLICATION IN VIVO, ESPECIALLY THROUGH THE SKIN IDEA AG (DE) 2004-04-22 WO claimed
US-6383471-B1 DRUG DELIVERY LIPOCINE, INC. 2002-05-07 US claimed
EP-1165048-A1 COMPOSITIONS AND METHODS FOR IMPROVED DELIVERY OF IONIZABLE HYDROPHOBIC THERAPEUTIC AGENTS Lipocine, Inc. (US) 2002-01-02 EP claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000059475-A1 COMPOSITIONS AND METHODS FOR IMPROVED DELIVERY OF IONIZABLE HYDROPHOBIC THERAPEUTIC AGENTS LIPOCINE, INC. (US) 2000-10-12 WO claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed
US-20260085062-A1 NOVEL COMPOUNDS AS CK2 INHIBITORS CAMBRIDGE ENTPR LTD (GB) 2026-03-26 US disclosed
US-4128641-A 2-METHYL-1,2,3,4,10,14B-HEXAHYDROPYRAZINO(1,2-A)DIBENZ-(C,F)AZEPINE HZI RESEARCH CENTER INC. (US) 1978-12-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260085062-A1 NOVEL COMPOUNDS AS CK2 INHIBITORS CSNK1A1, CSNK1G1, CSNK2A3 TSHR 3219/4885CHRM2 974/4885ADRA2A 1189/4885
US-20040105881-A1 Aggregates with increased deformability, comprising at least three amphipats, for improved transport through semi-permeable barriers and for the non-invasive drug application in vivo, especially through the skin CUTA, ABCG2, PIGS TSHR 3410/4885CHRM2 2986/4885ADRA2A 516/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.