SCHEMBL9449807

SCHEMBL9449807

CN1C[S+]([O-])c2cc(CCN3CCN(c4ncccn4)CC3)ccc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.46
HTR1A P08908 3/20 0.46
DRD3 P35462 2/20 0.46
DRD1 P21728 1/20 0.46
DRD5 P21918 1/20 0.46
HTR2A P28223 1/20 0.46
ABCB1 P08183 3/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
ALDH1A1 P00352 3/20 0.42
KDM4E B2RXH2 2/20 0.42
GAA P10253 1/20 0.42
USP2 O75604 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
ADRA2A P08913 1/20 0.42
CYP2D6 P10635 1/20 0.42
ADRA2B P18089 1/20 0.42
ADRA2C P18825 1/20 0.42
NFKB1 P19838 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9449641 0.88 ADRA1D (0.51) DRD2HTR1ADRD3DRD1DRD5
SCHEMBL9449660 0.83 HTR1A (0.47) DRD2HTR1ADRD3HTR2A
SCHEMBL8785466 0.81 DRD2 (0.46) DRD2HTR1ADRD3DRD1DRD5
SCHEMBL7759823 0.80 SIGMAR1 (0.48) DRD2HTR1AKMT2AADRA1AKCNH2
Hydrochloric Acid SCHEMBL9449928 0.80 HTR1A (0.51) DRD2HTR1ADRD3DRD1DRD5
SCHEMBL9449597 0.79 SIGMAR1 (0.55) HTR1AKDM4EGAACYP1A2CYP2D6
Hydrochloric Acid SCHEMBL9449688 0.78 ADRA1D (0.61) DRD2HTR1ADRD1HTR2AADRA1A
Hydrochloric Acid SCHEMBL9437976 0.76 HTR1A (0.60) DRD2HTR1AHTR2AABCB1ALDH1A1
SCHEMBL7756765 0.76 SIGMAR1 (0.58) HTR1ACYP1A2CYP2D6
SCHEMBL8109164 0.75 SIGMAR1 (0.51) DRD2MEN1KMT2ACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5234924-A Hypotensive agents ADIR ET COMPAGNIE (FR) 1993-08-10 US claimed