SCHEMBL9450889

SCHEMBL9450889

Cc1cccc(Cl)c1OC1CN(C(=O)N(C)C)C1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 7/20 0.40
HTR1A P08908 1/20 0.39
SLC6A2 P23975 1/20 0.39
OXTR P30559 3/20 0.38
AVPR1A P37288 2/20 0.38
POLB P06746 1/20 0.37
DRD2 P14416 2/20 0.37
DRD3 P35462 2/20 0.37
PDE9A O76083 1/20 0.37
USP30 Q70CQ3 1/20 0.36
RORC P51449 1/20 0.35
KDM4E B2RXH2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9450761 0.85 HTR1A (0.41) HTR1ASLC6A2POLBPDE9AKDM4E
SCHEMBL9450885 0.84 HTR1A (0.43) HTR1ASLC6A2POLBPDE9AKDM4E
SCHEMBL9450786 0.82 SCN9A (0.41) HTR1ASLC6A2POLBPDE9A
SCHEMBL9683890 0.74 ALDH1A1 (0.43) KIF11HTR1ASLC6A2KDM4E
SCHEMBL9733010 0.72 RBP4 (0.50) KIF11OXTRAVPR1ARORCKDM4E
SCHEMBL9450752 0.69 SLC6A2 (0.40) HTR1ASLC6A2DRD3PDE9A
SCHEMBL9354245 0.68 OXTR (0.48) KIF11OXTRAVPR1A
SCHEMBL9450789 0.68 POLB (0.37) HTR1ASLC6A2POLBKDM4E
SCHEMBL5363791 0.67 HTR1A (0.58) HTR1ASLC6A2
SCHEMBL10609153 0.67 SCD (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0560905-A1 3-[2-CHLORO-4-(TRIFLUOROMETHYL)PHENOXY]-1-AZETIDINE CARBOXAMIDES HAVING ANTICONVULSANT ACTIVITY. ROBINS CO INC A H (US) 1993-09-22 EP disclosed
WO-1992010474-A1 3-[2-CHLORO-4-(TRIFLUOROMETHYL)PHENOXY]-1-AZETIDINE CARBOXAMIDES HAVING ANTICONVULSANT ACTIVITY A.H. ROBINS COMPANY, INCORPORATED (US) 1992-06-25 WO disclosed
US-5095014-A 3-(2-chloro-4-(trifluoromethyl)phenoxy)-1-azetidine carboxamides having anticonvulsant activity A. H. ROBINS COMPANY, INCORPORATED (US) 1992-03-10 US disclosed