SCHEMBL9459228

SCHEMBL9459228

Cc1ccccc1CC(CS)NC(=O)c1ccncc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTRB1 P17538 1/20 0.53
ECE1 P42892 2/20 0.51
ROCK1 Q13464 7/20 0.48
ROCK2 O75116 6/20 0.48
PRKG1 Q13976 6/20 0.48
PKN2 Q16513 6/20 0.48
CLK4 Q9HAZ1 6/20 0.48
RPS6KA5 O75582 5/20 0.48
GSK3B P49841 5/20 0.48
PRKACA P17612 4/20 0.48
PRKX P51817 4/20 0.48
MAPK1 P28482 4/20 0.48
GSK3A P49840 4/20 0.48
SGK2 Q9HBY8 4/20 0.48
IRAK1 P51617 4/20 0.48
RPS6KA4 O75676 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.47
PRKG2 Q13237 5/20 0.43
RPS6KB1 P23443 4/20 0.43
AKT1 P31749 4/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9458948 0.86 CTRB1 (0.58) CTRB1ECE1ROCK1ROCK2PRKG1
SCHEMBL9459397 0.83 L3MBTL1 (0.43) ROCK1ROCK2PRKG1PKN2CLK4
SCHEMBL9486724 0.80 CTRB1 (0.54) CTRB1ECE1ALDH1A1HPGDKMT2A
SCHEMBL7357606 0.80 CTRB1 (0.54) CTRB1ECE1ALDH1A1HPGDKMT2A
SCHEMBL9458824 0.78 CTRB1 (0.49) CTRB1ECE1ALDH1A1HPGD
SCHEMBL9459389 0.78 HTT (0.57) CTRB1ECE1ALDH1A1HPGD
SCHEMBL12518290 0.75 CTSL (0.44) ROCK1ROCK2PRKG1PKN2CLK4
SCHEMBL30780061 0.74 HPGD (0.77) ROCK1ROCK2PRKG1PKN2CLK4
SCHEMBL1568387 0.74 HPGD (0.77) ROCK1ROCK2PRKG1PKN2CLK4
SCHEMBL9322253 0.72 CTRB1 (0.53) CTRB1ECE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5232920-A For treating hypertension and congestive heart failure in mammals SCHERING CORPORATION (US) 1993-08-03 US disclosed