SCHEMBL9483544

SCHEMBL9483544

CC(=O)Oc1ccc(C[C@H](NC(=O)OCc2ccccc2)C(=O)N2CCCN(CCCc3ccccc3)CC2)cc1

nearest known ligand 0.59

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 4/20 0.59
ITGA2B P08514 4/20 0.59
P2RX7 Q99572 14/20 0.51
HRH2 P25021 1/20 0.48
HRH1 P35367 1/20 0.48
OPRK1 P41145 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9483363 0.90 ITGB3 (0.59) ITGB3ITGA2BP2RX7OPRK1
SCHEMBL9483220 0.83 P2RX7 (0.69) P2RX7
SCHEMBL9484405 0.82 ITGB3 (0.55) ITGB3ITGA2BP2RX7
SCHEMBL9819722 0.80 ITGB3 (0.52) ITGB3ITGA2BOPRK1
SCHEMBL8750802 0.80 TACR1 (0.60) ITGB3ITGA2BP2RX7OPRK1
SCHEMBL8750811 0.80 TACR1 (0.60) ITGB3ITGA2BP2RX7OPRK1
SCHEMBL11257249 0.78 TACR1 (0.63) P2RX7
SCHEMBL11257246 0.78 TACR1 (0.63) P2RX7
SCHEMBL11232416 0.77 ITGB3 (0.62) ITGB3ITGA2BP2RX7
SCHEMBL9634993 0.73 P2RX7 (0.69) P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5245034-A Compound having vessel smooth muscle relaxation activity Hidaka, Kiroyoshi (JP) 1993-09-14 US disclosed
US-5216150-A Muscle relaxant; enzyme inhibitor and platelet aggutination inhibitor Hidaka, Hiroyoshi (JP) 1993-06-01 US disclosed