SCHEMBL9483363

SCHEMBL9483363

O=C(N[C@@H](Cc1ccc(O)cc1)C(=O)N1CCCN(CCCc2ccccc2)CC1)OCc1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 4/20 0.59
ITGA2B P08514 4/20 0.59
MC4R P32245 1/20 0.53
P2RX7 Q99572 7/20 0.49
CTSL P07711 2/20 0.48
CTSB P07858 2/20 0.48
CTSK P43235 1/20 0.48
FNTA P49354 1/20 0.48
FNTB P49356 1/20 0.48
OPRK1 P41145 2/20 0.47
CHRM3 P20309 1/20 0.47
PRSS1 P07477 1/20 0.47
PRSS2 P07478 1/20 0.47
PRSS3 P35030 1/20 0.47
TPSAB1 Q15661 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9483544 0.90 ITGB3 (0.59) ITGB3ITGA2BP2RX7OPRK1
SCHEMBL9819722 0.85 ITGB3 (0.52) ITGB3ITGA2BOPRK1CHRM3PRSS1
SCHEMBL8750802 0.84 TACR1 (0.60) ITGB3ITGA2BP2RX7CTSLCTSB
SCHEMBL8750811 0.84 TACR1 (0.60) ITGB3ITGA2BP2RX7CTSLCTSB
SCHEMBL11257249 0.82 TACR1 (0.63) P2RX7CTSLCTSBCTSK
SCHEMBL11257246 0.82 TACR1 (0.63) P2RX7CTSLCTSBCTSK
SCHEMBL9634993 0.81 P2RX7 (0.69) MC4RP2RX7
SCHEMBL9484550 0.81 OPRK1 (0.67) OPRK1CHRM3
SCHEMBL9484534 0.81 OPRK1 (0.67) OPRK1CHRM3
SCHEMBL9483704 0.81 MC4R (0.61) MC4RP2RX7CTSLCTSBCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5245034-A Compound having vessel smooth muscle relaxation activity Hidaka, Kiroyoshi (JP) 1993-09-14 US disclosed
US-5216150-A Muscle relaxant; enzyme inhibitor and platelet aggutination inhibitor Hidaka, Hiroyoshi (JP) 1993-06-01 US disclosed
US-5081246-A Isoquinolino sulfonamino derivatives Hidaka, Hiroyoshi (JP) 1992-01-14 US disclosed