SCHEMBL9507241

SCHEMBL9507241

COc1ccc(C(S)c2c(CC(CC(C)C)(C(=O)O)C(=O)O)cccc2C(F)(F)F)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 1/20 0.41
AKR1C4 P17516 1/20 0.37
AKR1C3 P42330 1/20 0.37
AKR1C2 P52895 1/20 0.37
AKR1C1 Q04828 1/20 0.37
BMP1 P13497 1/20 0.37
MEN1 O00255 4/20 0.37
KMT2A Q03164 4/20 0.37
GAA P10253 2/20 0.36
CMA1 P23946 2/20 0.36
ALDH1A1 P00352 3/20 0.36
KDM4E B2RXH2 1/20 0.36
HTT P42858 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
LMNA P02545 1/20 0.35
ATM Q13315 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
LNPEP Q9UIQ6 1/20 0.35
MAOB P27338 1/20 0.34
NPC1 O15118 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9510979 0.77 MMP1 (0.42) MMP1BMP1MEN1KMT2AGAA
SCHEMBL9509591 0.65 FFAR1 (0.39) MMP1GAAL3MBTL1
SCHEMBL9510871 0.63 ALDH1A1 (0.40) MMP1MEN1KMT2AGAAALDH1A1
SCHEMBL9511010 0.63 IDO1 (0.42) MMP1MEN1KMT2A
Anisole SCHEMBL7204405 0.61 CA4 (0.50) ALDH1A1
SCHEMBL9507230 0.61 CTSB (0.40) MEN1KMT2AGAAALDH1A1HTT
SCHEMBL7314497 0.61 AKR1C3 (0.40) AKR1C4AKR1C3AKR1C2AKR1C1MEN1
SCHEMBL2433696 0.59 ACP3 (0.56) KMT2AALDH1A1TDP1L3MBTL1NPC1
SCHEMBL7948715 0.58 CA1 (0.58) GAAALDH1A1KDM4ETDP1L3MBTL1
SCHEMBL5208103 0.58 LDHA (0.55) ALDH1A1KDM4EHTTLMNANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0358305-B1 MERCAPTO-PHENYLALCANOYLAMINO ACID AMIDES, THEIR PREPARATION AND THEIR USE AS COLLAGENASE INHIBITORS BEECHAM GROUP PLC (GB) 1993-08-25 EP disclosed
US-5124322-A Antiarthritic agents BEECHAM GROUP P.L.C. (GB) 1992-06-23 US disclosed
EP-0358305-A1 Mercapto-phenylalcanoylamino acid amides, their preparation and their use as collagenase inhibitors BEECHAM GROUP PLC (GB) 1990-03-14 EP disclosed