SCHEMBL951718

SCHEMBL951718

NC(=O)CCCc1cccc(-c2cn[nH]c2)c1

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 14/20 0.50
ROCK1 Q13464 5/20 0.50
AKT2 P31751 2/20 0.47
CTSV O60911 1/20 0.43
CTSL P07711 1/20 0.43
CTSB P07858 1/20 0.43
CTSS P25774 1/20 0.43
CHEK1 O14757 3/20 0.43
AKT1 P31749 1/20 0.42
CHEK2 O96017 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL934607 0.78 EPHX2 (0.51)
SCHEMBL13737919 0.77 GRIN2D (0.56) ROCK2ROCK1AKT2CTSVCTSL
SCHEMBL933474 0.77 PRKCI (0.57) ROCK2
SCHEMBL952139 0.77 CD74 (0.54) CTSVCTSLCTSBCTSS
SCHEMBL951716 0.76 CTSV (0.52) ROCK2ROCK1CTSVCTSLCTSB
SCHEMBL5218911 0.74 TBXAS1 (0.55)
SCHEMBL22501830 0.74 ROCK2 (0.59) ROCK2ROCK1CTSVCTSLCTSB
SCHEMBL6037977 0.74 MAPT (0.54)
SCHEMBL3663278 0.74 CCNT1 (0.52) ROCK2ROCK1AKT2CHEK1AKT1
SCHEMBL19837880 0.73 CHEK1 (0.50) ROCK2ROCK1CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011006935-A2 TETRAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2011-01-20 WO disclosed