SCHEMBL9750874

SCHEMBL9750874

C=C(C#N)c1c(-c2ccc(F)cc2)cn(C(C)C)c1C(C)C

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HMGCR P04035 5/20 0.41
TGFBR1 P36897 8/20 0.35
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32
TGFBR2 P37173 2/20 0.32
ABCB1 P08183 1/20 0.32
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
GAA P10253 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
MAPK13 O15264 1/20 0.30
MAPK12 P53778 1/20 0.30
MAPK11 Q15759 1/20 0.30
MAPK14 Q16539 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9751010 0.80 HMGCR (0.49) HMGCRTGFBR1ADORA2AADORA1TGFBR2
SCHEMBL9750803 0.79 HMGCR (0.49) HMGCRTGFBR1TGFBR2GAAMAPK13
SCHEMBL9732188 0.73 PKM (0.37) KDM4EALDH1A1SMN1; SMN2
SCHEMBL9518155 0.73 HMGCR (0.53) HMGCRTGFBR1ADORA2AADORA1TGFBR2
SCHEMBL9518177 0.72 HMGCR (0.47) HMGCR
SCHEMBL9750967 0.71 HMGCR (0.47) HMGCRABCB1KDM4EGAASMN1; SMN2
SCHEMBL9764350 0.70 KDM4E (0.43) HMGCRKDM4EALDH1A1
SCHEMBL9751046 0.69 HMGCR (0.55) HMGCRADORA2AADORA1ALDH1A1MAPK13
SCHEMBL9750986 0.68 ABCB1 (0.52) HMGCRABCB1KDM4EALDH1A1GAA
SCHEMBL9024316 0.68 PTGS2 (0.33) HMGCRKDM4EALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5055484-A Anticholesterol and antilipemic agent HOECHST AKTIENGESELLSCHAFT (DE) 1991-10-08 US disclosed