SCHEMBL9530704

SCHEMBL9530704

CSc1ccc(C2=CCN(CCC3OCCO3)CC2)cc1

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 12/20 0.40
HTR1D P28221 1/20 0.39
QDPR P09417 1/20 0.38
DRD2 P14416 2/20 0.37
DRD3 P35462 2/20 0.37
DRD4 P21917 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9529720 0.83 SIGMAR1 (0.57) SIGMAR1HTR1DDRD2
SCHEMBL9531082 0.83 SIGMAR1 (0.57) SIGMAR1DRD2
SCHEMBL9532157 0.82 SIGMAR1 (0.54) SIGMAR1HTR1D
SCHEMBL9533235 0.75 HTR1D (0.44) SIGMAR1HTR1DDRD2DRD4
SCHEMBL3318787 0.67 DRD2 (0.46) SIGMAR1DRD2DRD3DRD4
SCHEMBL23735080 0.66 KDM4E (0.39) SIGMAR1DRD2DRD4
SCHEMBL20182439 0.66 MEN1 (0.50) QDPR
Sulfuric Acid SCHEMBL17364146 0.65 SIGMAR1 (0.41) SIGMAR1DRD2DRD3DRD4
SCHEMBL466989 0.64 SIGMAR1 (0.57) SIGMAR1
SCHEMBL7303423 0.63 QDPR (0.51) SIGMAR1QDPRDRD2DRD3DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0556342-A1 NEW 1-AZABICYCLOALKANE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESS FOR PREPARING SAME GYOGYSZERKUTATO INTEZET K.V. (HU) 1993-08-25 EP disclosed
EP-0515548-A4 IMIDAZOLE ANGIOTENSIN II ANTAGONISTS INCORPORATING A SUBSTITUTED BENZYL ELEMENT 1993-03-10 EP disclosed
EP-0515548-A1 IMIDAZOLE ANGIOTENSIN II ANTAGONISTS INCORPORATING A SUBSTITUTED BENZYL ELEMENT MERCK & CO. INC. (US) 1992-12-02 EP disclosed
WO-1992007854-A1 NEW 1-AZABICYCLOALKANE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESS FOR PREPARING SAME GYÓGYSZERKUTATÓ INTÉZET KV. (HU) 1992-05-14 WO disclosed