SCHEMBL9530828

SCHEMBL9530828

c1ccc(N2CC(CN3CCN(c4cnccn4)CC3)Oc3ccccc32)cc1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.45
LMNA P02545 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
DRD4 P21917 2/20 0.44
GBA1 P04062 1/20 0.41
DRD2 P14416 2/20 0.41
DRD3 P35462 2/20 0.41
ADRA2A P08913 2/20 0.40
ADRA2B P18089 2/20 0.40
ADRA2C P18825 2/20 0.40
OPRM1 P35372 1/20 0.40
HTR1A P08908 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
SLC6A7 Q99884 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CASR P41180 1/20 0.39
ABCB1 P08183 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9529716 0.89 KCNH2 (0.50) DRD4DRD2ADRA2AADRA2BADRA2C
SCHEMBL9530044 0.84 ABCB1 (0.49) DRD4DRD2DRD3ADRA2AADRA2B
Hydrochloric Acid SCHEMBL10368330 0.82 ABCB1 (0.48) DRD4DRD2DRD3ADRA2AADRA2B
SCHEMBL10677091 0.82 ADRA2A (0.59) KDM4EGBA1DRD2ADRA2AADRA2B
SCHEMBL9696810 0.79 ADRA2A (0.59) ADRA2AADRA2BADRA2CHTR1ASIGMAR1
SCHEMBL9455117 0.78 CASR (0.45) LMNADRD4DRD2DRD3ADRA2A
SCHEMBL9455118 0.76 ADRA2A (0.70) DRD4DRD2DRD3ADRA2AADRA2B
SCHEMBL9529266 0.76 DRD2 (0.53) LMNADRD4DRD2HTR1ASIGMAR1
SCHEMBL9530260 0.75 SIGMAR1 (0.53) DRD4DRD2ADRA2AADRA2BADRA2C
SCHEMBL9530838 0.72 L3MBTL1 (0.46) KDM4ELMNAL3MBTL1DRD4OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0359790-B1 1,4-BENZOXAZINE AND 1,4-BENZOTHIAZINE DERIVATIVES AND PROCESS FOR THEIR PREPARATION ERBA CARLO SPA (IT) 1993-11-03 EP disclosed
US-5084454-A Tranquilizers and antinausea drugs FARMITALIA CARLO ERBA S.R.L. (IT) 1992-01-28 US disclosed