SCHEMBL9534814

SCHEMBL9534814

Cc1ccc2sc(CNC(=O)OCc3ccccc3)c3c2c1CCN(C)C3

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.42
ADRA2B P18089 1/20 0.42
ADRA2C P18825 1/20 0.42
ADRA1D P25100 1/20 0.42
ADRA1A P35348 1/20 0.42
ADRA1B P35368 1/20 0.42
ADORA1 P30542 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.40
TMEM97 Q5BJF2 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
PTGDR2 Q9Y5Y4 2/20 0.37
LMNA P02545 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9535094 0.84 ALDH1A1 (0.44) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL9535666 0.82 ADRA2A (0.41) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL9533677 0.72 ADRA2A (0.42) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL9535778 0.70 KAT2B (0.39) ADORA1TMEM97SIGMAR1KEAP1NFE2L2
SCHEMBL9533309 0.69 ADRA1D (0.68) ADRA2AADRA2BADRA2CADRA1DADRA1A
Benzyl Benzylcarbamate SCHEMBL1136818 0.64 PLAU (0.70) KEAP1NFE2L2LMNASMN1; SMN2ALDH1A1
Benzyl Benzylcarbamate SCHEMBL19810513 0.63 PLAU (0.68) KEAP1NFE2L2LMNASMN1; SMN2ALDH1A1
Benzyl Benzylcarbamate SCHEMBL9998166 0.63 PLAU (0.68) KEAP1NFE2L2LMNASMN1; SMN2ALDH1A1
Benzyl Benzylcarbamate SCHEMBL28413454 0.63 PLAU (0.68) KEAP1NFE2L2LMNASMN1; SMN2ALDH1A1
SCHEMBL12203724 0.62 SMN1; SMN2 (0.66) L3MBTL1NPC1RAB9ALMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0384677-B1 Alpha-adrenergic receptor antagonists SMITHKLINE BEECHAM CORP (US) 1993-12-01 EP disclosed
US-4981848-A CARDIOVASCULAR, HYPOTENSIVE, ANTIDEPRESSANT SMITHKLINE BEECHAM CORPORATION (US) 1991-01-01 US disclosed