SCHEMBL9540183

SCHEMBL9540183

O=c1[nH]c2ccccc2c(=O)n1CCN1CCC(Cc2nc3ccccc3n2Cc2cscn2)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.47
ALDH1A1 P00352 2/20 0.43
CYP3A4 P08684 2/20 0.43
HPGD P15428 2/20 0.43
CYP2C19 P33261 2/20 0.43
SLC6A3 Q01959 2/20 0.43
SLC18A2 Q05940 2/20 0.43
DRD2 P14416 2/20 0.43
ADRA2B P18089 2/20 0.43
DRD3 P35462 2/20 0.43
MEN1 O00255 1/20 0.43
LMNA P02545 1/20 0.43
CYP1A2 P05177 1/20 0.43
HTR1A P08908 1/20 0.43
MAPT P10636 1/20 0.43
CYP2C9 P11712 1/20 0.43
ADRA2C P18825 1/20 0.43
DRD1 P21728 1/20 0.43
DRD4 P21917 1/20 0.43
HTR1D P28221 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9538362 0.84 ACHE (0.48) ACHEALDH1A1CYP3A4HPGDCYP2C19
SCHEMBL9537087 0.83 TSHR (0.54) ACHEALDH1A1CYP3A4HPGDCYP2C19
SCHEMBL9537175 0.81 HRH1 (0.53) ALDH1A1CYP2C19DRD2DRD3MEN1
SCHEMBL9536342 0.80 ALDH1A1 (0.50) ALDH1A1CYP2C19MEN1LMNACYP1A2
SCHEMBL10550233 0.79 ACHE (0.51) ACHEALDH1A1CYP3A4HPGDCYP2C19
SCHEMBL10551946 0.78 TSHR (0.52) ACHEALDH1A1CYP3A4HPGDCYP2C19
SCHEMBL9539219 0.76 HRH1 (0.42) ALDH1A1DRD2DRD3MEN1LMNA
SCHEMBL9537082 0.76 HTR2A (0.56) ALDH1A1CYP3A4HPGDCYP2C19SLC6A3
SCHEMBL9536214 0.75 SLC18A2 (0.53) ACHEALDH1A1CYP3A4HPGDCYP2C19
SCHEMBL9539277 0.75 ALDH1A1 (0.49) ALDH1A1CYP3A4HPGDDRD2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP claimed