SCHEMBL9538362

SCHEMBL9538362

O=c1[nH]c2ccccc2c(=O)n1CCN1CCC(Cc2nc3ccccc3n2Cc2cccs2)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.48
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
SLC6A9 P48067 1/20 0.45
SLC18A2 Q05940 3/20 0.45
ALDH1A1 P00352 2/20 0.44
CYP3A4 P08684 2/20 0.44
HPGD P15428 2/20 0.44
CYP2C19 P33261 2/20 0.44
SLC6A3 Q01959 2/20 0.44
LMNA P02545 1/20 0.44
CYP1A2 P05177 1/20 0.44
HTR1A P08908 1/20 0.44
MAPT P10636 1/20 0.44
CYP2C9 P11712 1/20 0.44
DRD2 P14416 1/20 0.44
ADRA2B P18089 1/20 0.44
ADRA2C P18825 1/20 0.44
DRD1 P21728 1/20 0.44
DRD4 P21917 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9537087 0.85 TSHR (0.54) ACHEMEN1KMT2ASLC18A2ALDH1A1
SCHEMBL9540183 0.84 ACHE (0.47) ACHEMEN1KMT2ASLC18A2ALDH1A1
SCHEMBL10551946 0.81 TSHR (0.52) ACHEMEN1KMT2ASLC18A2ALDH1A1
SCHEMBL10550233 0.80 ACHE (0.51) ACHEMEN1KMT2ASLC18A2ALDH1A1
SCHEMBL9539084 0.79 MEN1 (0.52) MEN1KMT2ASLC6A9ALDH1A1HPGD
SCHEMBL9539277 0.78 ALDH1A1 (0.49) MEN1KMT2AALDH1A1CYP3A4HPGD
SCHEMBL9537082 0.77 HTR2A (0.56) MEN1KMT2ASLC18A2ALDH1A1CYP3A4
SCHEMBL10549103 0.76 SLC18A2 (0.53) ACHEMEN1KMT2ASLC18A2ALDH1A1
SCHEMBL9537145 0.75 SLC6A9 (0.53) MEN1KMT2ASLC6A9HPGDMAPT
SCHEMBL9534954 0.75 SMN1; SMN2 (0.52) SLC6A9ALDH1A1CYP3A4HPGDCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP claimed