SCHEMBL9537865

SCHEMBL9537865

FC(F)(F)c1cccc(N2CCN(CCSc3nc[nH]n3)CC2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.53
DRD2 P14416 6/20 0.52
HTR1A P08908 5/20 0.50
ALDH1A1 P00352 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
MAPT P10636 1/20 0.50
TSHR P16473 1/20 0.50
NFKB1 P19838 1/20 0.50
MAPK1 P28482 1/20 0.50
CYP2C19 P33261 1/20 0.50
THPO P40225 1/20 0.50
MTOR P42345 1/20 0.50
BLM P54132 1/20 0.50
PMP22 Q01453 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
HTR7 P34969 1/20 0.50
HTR2A P28223 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7674560 0.77 DRD2 (0.62) SIGMAR1DRD2HTR1AHTR7HTR2A
SCHEMBL12468893 0.77 SIGMAR1 (0.53) SIGMAR1DRD2HTR1AALDH1A1CYP1A2
SCHEMBL9535966 0.76 MAPT (0.45) DRD2HTR1AMAPTHTR2A
SCHEMBL11465528 0.75 SIGMAR1 (0.76) SIGMAR1DRD2HTR1AALDH1A1CYP1A2
SCHEMBL9538643 0.74 KDM4E (0.45) SIGMAR1DRD2HTR1AALDH1A1CYP2D6
SCHEMBL4608279 0.73 DRD2 (0.53) SIGMAR1DRD2HTR1AHTR7HTR2A
SCHEMBL1253143 0.73 SIGMAR1 (0.69) SIGMAR1DRD2HTR1AALDH1A1CYP1A2
Hydrochloric Acid SCHEMBL7323720 0.73 HTR1A (0.53) SIGMAR1HTR1AALDH1A1CYP1A2CYP3A4
SCHEMBL12469526 0.73 NPSR1 (0.63) SIGMAR1DRD2HTR1AALDH1A1CYP1A2
SCHEMBL9537473 0.73 KDM4E (0.46) DRD2HTR1AALDH1A1HTR2AADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0254623-B1 AMINOALKYLTHIO TRIAZOLOPYRIDINE OR TRIAZOLOQUINOLINE DERIVATIVES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS CONTAINING THEM, PARTICULARLY USEFUL AS ANTALGICS LABORATOIRES UPSA (FR) 1993-06-09 EP disclosed
EP-0254623-A1 Aminoalkylthio triazolopyridine or triazoloquinoline derivatives, process for their preparation, medicaments containing them, particularly useful as antalgics LABORATOIRES UPSA (FR) 1988-01-27 EP disclosed