SCHEMBL9538643

SCHEMBL9538643

Fc1ccccc1N1CCN(CCSc2nc[nH]n2)CC1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.45
ALDH1A1 P00352 2/20 0.45
POLB P06746 1/20 0.45
TSHR P16473 1/20 0.45
DRD2 P14416 2/20 0.45
ADRA1A P35348 1/20 0.45
DRD3 P35462 1/20 0.45
DAO P14920 1/20 0.44
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
DRD4 P21917 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
HTR1A P08908 1/20 0.42
HTR2A P28223 1/20 0.42
HTR7 P34969 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9537473 0.87 KDM4E (0.46) KDM4EALDH1A1DRD2ADRA1ALMNA
SCHEMBL28070630 0.86 ADRA1B (0.46) DRD2ADRA1ADRD3SIGMAR1HTR1A
SCHEMBL9535969 0.86 AR (0.48) ALDH1A1DRD2ADRA1ADRD3LMNA
SCHEMBL9540523 0.81 HTR1A (0.48) ALDH1A1POLBDRD2DRD3MAPT
SCHEMBL9535966 0.76 MAPT (0.45) DRD2MAPTDRD4HTR1AHTR2A
SCHEMBL9537865 0.74 SIGMAR1 (0.53) ALDH1A1TSHRDRD2ADRA1ADRD3
SCHEMBL9536766 0.74 ALDH1A1 (0.42) KDM4EALDH1A1POLBTSHRDRD2
SCHEMBL9535704 0.72 KDM4E (0.59) KDM4EALDH1A1DRD2DRD3LMNA
SCHEMBL10646895 0.71 DRD2 (0.49) DRD2DRD3SIGMAR1HTR1AHTR2A
SCHEMBL4256755 0.70 KDM4E (0.63) KDM4EALDH1A1POLBTSHRDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0254623-B1 AMINOALKYLTHIO TRIAZOLOPYRIDINE OR TRIAZOLOQUINOLINE DERIVATIVES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS CONTAINING THEM, PARTICULARLY USEFUL AS ANTALGICS LABORATOIRES UPSA (FR) 1993-06-09 EP disclosed