SCHEMBL9541838

SCHEMBL9541838

FC(F)(F)c1cc(C=P(c2ccccc2)(c2ccccc2)c2ccccc2)cc(C(F)(F)F)c1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.44
TDO2 P48775 2/20 0.44
ALDH1A1 P00352 1/20 0.41
TSHR P16473 1/20 0.41
P2RX1 P51575 1/20 0.37
MAPT P10636 3/20 0.36
KDM4E B2RXH2 2/20 0.36
KIF11 P52732 1/20 0.36
FBP1 P09467 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
TACR1 P25103 4/20 0.34
NFE2L2 Q16236 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MAOB P27338 1/20 0.33
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9540307 0.86 FBP1 (0.47) IDO1TDO2ALDH1A1TSHRMAPT
SCHEMBL9539528 0.83 ALDH1A1 (0.48) ALDH1A1TSHRKIF11FBP1NPC1
SCHEMBL9538889 0.73 NPBWR1 (0.40) ALDH1A1TSHRMAPTKDM4EKIF11
SCHEMBL1132385 0.73 ALDH1A1 (0.39) ALDH1A1TSHRMAPTFBP1MEN1
SCHEMBL3593834 0.71 HSP90AA1 (0.49) ALDH1A1P2RX1MAPTTACR1NPC1
SCHEMBL9538666 0.71 NPBWR1 (0.39) ALDH1A1TSHRMAPTKIF11MEN1
Fluoride SCHEMBL27260416 0.71 ALDH1A1 (0.38) ALDH1A1TSHRMAPTFBP1MEN1
SCHEMBL5249757 0.70 CES2 (0.44) IDO1TDO2ALDH1A1TSHRMAPT
SCHEMBL7616716 0.69 P2RX1 (0.46) ALDH1A1TSHRP2RX1KIF11TACR1
SCHEMBL9541494 0.68 NFE2L2 (0.52) ALDH1A1TSHRMAPTFBP1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0311955-B1 BICYCLIC PEROXIDE F. HOFFMANN-LA ROCHE AG (CH) 1993-04-21 EP disclosed
US-5134240-A Malaria therapy HOFFMANN-LAROCHE, INC. (US) 1992-07-28 US disclosed
US-4977184-A Bicyclic peroxides compositions for and treatment of malaria therewith HOFFMANN-LA ROCHE INC. (US) 1990-12-11 US disclosed
EP-0311955-A2 Bicyclic peroxide F. HOFFMANN-LA ROCHE AG (CH) 1989-04-19 EP disclosed