SCHEMBL9540523

SCHEMBL9540523

Fc1ccc(N2CCN(CCSc3nc[nH]n3)CC2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 7/20 0.48
DRD2 P14416 7/20 0.48
HTR2A P28223 7/20 0.48
DRD3 P35462 7/20 0.48
DRD1 P21728 3/20 0.47
DRD5 P21918 3/20 0.47
SLC6A3 Q01959 3/20 0.46
HRH1 P35367 4/20 0.44
SIGMAR1 Q99720 3/20 0.44
TMEM97 Q5BJF2 2/20 0.44
HTR2C P28335 1/20 0.44
SLC6A2 P23975 4/20 0.44
SLC6A4 P31645 4/20 0.44
HRH2 P25021 1/20 0.43
HRH3 Q9Y5N1 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9535966 0.88 MAPT (0.45) HTR1ADRD2HTR2AHTR2CMEN1
SCHEMBL10646895 0.81 DRD2 (0.49) HTR1ADRD2HTR2ADRD3DRD1
SCHEMBL9538643 0.81 KDM4E (0.45) HTR1ADRD2HTR2ADRD3SIGMAR1
SCHEMBL9537865 0.78 SIGMAR1 (0.53) HTR1ADRD2HTR2ADRD3DRD1
SCHEMBL9537473 0.77 KDM4E (0.46) HTR1ADRD2HTR2ADRD1SLC6A3
SCHEMBL9537905 0.76 SIGMAR1 (0.47) HTR1ADRD2HTR2ASIGMAR1MEN1
SCHEMBL9535969 0.76 AR (0.48) HTR1ADRD2HTR2ADRD3HTR2C
SCHEMBL9536766 0.76 ALDH1A1 (0.42) DRD2DRD3HRH1SIGMAR1HRH2
SCHEMBL9536717 0.71 HTR1A (0.38) HTR1ADRD2HTR2ADRD3DRD1
SCHEMBL8011318 0.70 DRD2 (0.69) HTR1ADRD2HTR2ADRD3DRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0254623-B1 AMINOALKYLTHIO TRIAZOLOPYRIDINE OR TRIAZOLOQUINOLINE DERIVATIVES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS CONTAINING THEM, PARTICULARLY USEFUL AS ANTALGICS LABORATOIRES UPSA (FR) 1993-06-09 EP disclosed