Bromide

Bromide

SCHEMBL9545828

Br.Cc1cccc(COc2ccc(C3(C)OC(=O)N(Nc4ccccc4)C3=N)cc2)c1

nearest known ligand 0.42

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ACHE known ✓ P22303 1/20 0.39
MAOB P27338 8/20 0.42
NR1H4 Q96RI1 2/20 0.42
SIRT1 Q96EB6 2/20 0.41
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
FFAR1 O14842 2/20 0.39
MAOA P21397 2/20 0.38
MMP2 P08253 1/20 0.38
MMP13 P45452 1/20 0.38
GRM5 P41594 1/20 0.37
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9545818 0.90 MAOB (0.44) MAOBNR1H4SIRT1OPRM1OPRD1
Bromide SCHEMBL8633989 0.80 MMP2 (0.39) SIRT1MMP2MMP13MAPT
SCHEMBL8637040 0.79 MMP2 (0.40) SIRT1MMP2MMP13MAPT
SCHEMBL8893376 0.75 SIRT1 (0.41) MAOBSIRT1MMP2MMP13MAPT
SCHEMBL9545815 0.73 MAOB (0.42) MAOBSIRT1OPRM1OPRD1ACHE
SCHEMBL9231335 0.73 NR1H4 (0.41) MAOBNR1H4SIRT1OPRM1OPRD1
SCHEMBL9207805 0.73 RAB9A (0.40) MAOBSIRT1ACHEFFAR1MAOA
SCHEMBL8892271 0.71 LMNA (0.52) MAPT
SCHEMBL8902452 0.70 SIRT1 (0.39) SIRT1MMP2MMP13MAPT
SCHEMBL9202236 0.69 SIRT1 (0.37) SIRT1MMP2MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993022299-A1 FUNGICIDAL OXAZOLIDINONES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1993-11-11 WO disclosed