SCHEMBL9564931

SCHEMBL9564931

CC(CC(C(=O)N(C)C)(c1ccccc1)c1ccccc1)N1CCC(Nc2nc3cncnc3n2Cc2ccco2)CC1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.34
TSHR P16473 6/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
MAPT P10636 5/20 0.33
NPSR1 Q6W5P4 3/20 0.33
KDM4E B2RXH2 3/20 0.33
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
GLA P06280 2/20 0.33
GAA P10253 1/20 0.33
RUNX1 Q01196 1/20 0.33
MCL1 Q07820 1/20 0.33
CBFB Q13951 1/20 0.33
LMNA P02545 5/20 0.33
HTT P42858 2/20 0.32
OPRM1 P35372 1/20 0.32
HSD17B10 Q99714 1/20 0.32
CACNA2D1 P54289 1/20 0.32
MAPK1 P28482 1/20 0.32
ADORA3 P0DMS8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9565024 0.90 LMNA (0.32) LMNA
SCHEMBL9565015 0.88 CHRM2 (0.35) MEN1KMT2ALMNAOPRM1
SCHEMBL9564816 0.76 NOS2 (0.46) ALDH1A1TSHRSMN1; SMN2MAPTKDM4E
SCHEMBL9866590 0.75 OPRM1 (0.43) ALDH1A1TSHRSMN1; SMN2NPSR1KDM4E
SCHEMBL8207942 0.73 KCNH2 (0.47) ALDH1A1SMN1; SMN2MAPTMEN1KMT2A
SCHEMBL9564789 0.73 NR4A2 (0.42) ALDH1A1TSHRMAPTKDM4EMEN1
SCHEMBL9564775 0.72 OPRM1 (0.48) ALDH1A1TSHRSMN1; SMN2NPSR1MEN1
SCHEMBL9564925 0.72 CHRM2 (0.38) ALDH1A1SMN1; SMN2KDM4ELMNAOPRM1
Water SCHEMBL9564807 0.72 NR4A2 (0.42) ALDH1A1TSHRMAPTKDM4EMEN1
Water SCHEMBL9564806 0.72 NR4A2 (0.42) ALDH1A1TSHRMAPTKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5258380-A Antiallergens, antihistamines JANSSEN PHARMACEUTICA N.V. (BE) 1993-11-02 US disclosed
US-5041448-A Antiallergens JANSSEN PHARMACEUTICA N.V. (BE) 1991-08-20 US disclosed
EP-0206415-A2 (4-Piperidinylmethyl and -hetero)purines JANSSEN PHARMACEUTICA N.V. (BE) 1986-12-30 EP disclosed